SCHEMBL8844191

SCHEMBL8844191

N#Cc1ccccc1C1CCN(Cc2ccccc2)C1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
ALDH1A1 P00352 1/20 0.49
CNR2 P34972 1/20 0.48
SIGMAR1 Q99720 2/20 0.48
GRIN1 Q05586 1/20 0.48
GRIN2B Q13224 1/20 0.48
HRH3 Q9Y5N1 1/20 0.47
DRD2 P14416 1/20 0.47
BCHE P06276 1/20 0.47
BACE1 P56817 1/20 0.47
RET P07949 1/20 0.46
CHRM4 P08173 1/20 0.46
DRD4 P21917 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9731324 0.82 ACHE (0.47) ACHEHRH3BCHEBACE1RET
SCHEMBL8844616 0.80 ACHE (0.48) ACHECNR2HRH3BCHEBACE1
SCHEMBL4896796 0.78 MEN1 (0.54) ACHEMEN1KMT2AALDH1A1SIGMAR1
SCHEMBL4896785 0.78 MEN1 (0.54) ACHEMEN1KMT2AALDH1A1SIGMAR1
SCHEMBL14163184 0.78 DRD4 (0.54) MEN1KMT2AHRH3DRD2DRD4
SCHEMBL8844253 0.77 HRH3 (0.60) ACHEMEN1KMT2AHRH3DRD2
SCHEMBL8009313 0.75 DRD4 (0.49) MEN1KMT2ADRD2DRD4
SCHEMBL20140665 0.75 PROKR1 (0.50) MEN1KMT2AALDH1A1DRD4
SCHEMBL851805 0.75 S1PR5 (0.46) KMT2AALDH1A1DRD2CHRM4
SCHEMBL22755777 0.75 MEN1 (0.68) ACHEMEN1KMT2ASIGMAR1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622966-A BACTERICIDES TREATING INFECTIONS WARNER-LAMBERT COMPANY (US) 1997-04-22 US disclosed
US-5446044-A Bactericides WARNER-LAMBERT COMPANY (US) 1995-08-29 US disclosed
US-5384407-A Pyrrolidine compounds WARNER-LAMBERT COMPANY (US) 1995-01-24 US disclosed
US-5342844-A 7-substituted quinolones and naphthyridones as antibacterial agents WARNER-LAMBERT COMPANY (US) 1994-08-30 US disclosed
WO-1993016077-A1 7-SUBSTITUTED QUINOLONES AND NAPHTHYRIDONES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1993-08-19 WO disclosed
US-5221676-A 7-substituted quinolones and naphthyridones as antibacterial agents WARNER-LAMBERT COMPANY (US) 1993-06-22 US disclosed