SCHEMBL8848089

SCHEMBL8848089

NCCn1nc2c3c(c(Cl)ccc31)C(=O)c1cnccc1-2

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 12/20 0.46
CDC25B P30305 1/20 0.38
CSNK1A1 P48729 1/20 0.33
CSNK1D P48730 1/20 0.33
CSNK1E P49674 1/20 0.33
CSNK1G2 P78368 1/20 0.33
CSNK1G1 Q9HCP0 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
ECE1 P42892 1/20 0.32
MUS81 Q96NY9 1/20 0.32
TDP1 Q9NUW8 3/20 0.32
KDM4E B2RXH2 1/20 0.32
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.32
CASP1 P29466 1/20 0.32
BLM P54132 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8847987 0.93 TOP2A (0.45) TOP2ACDC25BCSNK1A1CSNK1DCSNK1E
SCHEMBL8847912 0.89 TOP2A (0.46) TOP2ACDC25BMAOAMAOBKDM4E
SCHEMBL10801104 0.86 TOP2A (0.54) TOP2ATDP1
SCHEMBL7817561 0.86 TOP2A (0.41) TOP2ACDC25BMAOAMAOBECE1
SCHEMBL7804662 0.86 TOP2A (0.48) TOP2ACDC25BTDP1KDM4ETP53
SCHEMBL7812061 0.84 TOP2A (0.45) TOP2ATDP1
SCHEMBL7814010 0.84 TOP2A (0.45) TOP2ACDC25BSMN1; SMN2
SCHEMBL7827886 0.84 TOP2A (0.36) TOP2ACDC25BMAOAMAOBKDM4E
SCHEMBL7804837 0.83 TOP2A (0.50) TOP2ACDC25BKDM4ETP53CYP3A4
SCHEMBL7820225 0.83 ECE1 (0.49) TOP2AMAOAMAOBECE1MUS81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5604246-A HAVING POTENCY AGAINST MULTIDRUG RESISTANT TUMORS BOEHRINGER MANNHEIM ITALIA SPA (IT) 1997-02-18 US disclosed
US-5519029-A ANTITUMOR AGENTS BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1996-05-21 US disclosed