SCHEMBL8848337

SCHEMBL8848337

CC(=O)/C(=C/c1cc(O)c(O)c([N+](=O)[O-])c1)c1ccc(C)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 3/20 0.64
ABCC3 O15438 2/20 0.59
ABCC4 O15439 2/20 0.59
ABCB11 O95342 2/20 0.59
COMT P21964 2/20 0.59
NR1I2 O75469 1/20 0.59
TTR P02766 1/20 0.59
NR3C1 P04150 1/20 0.59
PGR P06401 1/20 0.59
HTR1A P08908 1/20 0.59
ADORA3 P0DMS8 1/20 0.59
RARB P10826 1/20 0.59
SLC6A2 P23975 1/20 0.59
ADORA1 P30542 1/20 0.59
ADRA1A P35348 1/20 0.59
PTGS2 P35354 1/20 0.59
SLC6A3 Q01959 1/20 0.59
KCNH2 Q12809 1/20 0.59
KLF10 Q13118 1/20 0.59
PDE3A Q14432 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8848340 1.00 GPR35 (0.64) GPR35ABCC3ABCC4ABCB11COMT
SCHEMBL8848710 0.89 GPR35 (0.65) GPR35MEN1KMT2AALDH1A1MAPT
SCHEMBL8848706 0.89 GPR35 (0.65) GPR35MEN1KMT2AALDH1A1MAPT
Tolcapone SCHEMBL4391775 0.82 TTR (0.73) GPR35ABCC3ABCC4ABCB11COMT
SCHEMBL8848407 0.79 DBH (0.77) GPR35ABCC3ABCC4ABCB11COMT
SCHEMBL8848409 0.79 DBH (0.77) GPR35ABCC3ABCC4ABCB11COMT
Nitecapone SCHEMBL128420 0.78 GPR35 (1.00) GPR35ABCC3ABCC4ABCB11COMT
Nitecapone SCHEMBL7039409 0.78 GPR35 (1.00) GPR35ABCC3ABCC4ABCB11COMT
SCHEMBL7279188 0.78 GPR35 (0.78) GPR35ABCC3ABCC4ABCB11COMT
SCHEMBL7279195 0.78 GPR35 (0.78) GPR35ABCC3ABCC4ABCB11COMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0444899-B1 Catechol derivatives, their physiologically acceptable salts, esters and their use in the treatment of tissue damage induced by lipid peroxidation ORION YHTYMAE OY (FI) 1997-02-05 EP disclosed
US-5489614-A MEDICINAL ANTIOXIDANTS USED IN PREVENTION AND TREATMENT OF TISSUE DAMAGE INDUCED BY LIPID PEROXIDATION ORION-YHTYMA OY (FI) 1996-02-06 US disclosed
EP-0444899-A2 Catechol derivatives, their physiologically acceptable salts, esters and their use in the treatment of tissue damage induced by lipid peroxidation ORION-YHTYMÀ„ OY (FI) 1991-09-04 EP disclosed