SCHEMBL88501

SCHEMBL88501

CCOC(=O)/C(C)=C/C(C(C)C)N(C)C(=O)C(NC(=O)C1CCN(C)CC1)C(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 2/20 0.44
CTSB P07858 1/20 0.36
GAA P10253 3/20 0.35
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 4/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL58783 1.00 TUBB1 (0.44) TUBB1CTSBGAAHPGDSMN1; SMN2
SCHEMBL12201945 0.89 TUBB1 (0.52) TUBB1GAAHPGDSMN1; SMN2ALOX15
SCHEMBL58787 0.89 TUBB1 (0.52) TUBB1GAAHPGDSMN1; SMN2ALOX15
SCHEMBL14592518 0.89 TUBB1 (0.52) TUBB1GAAHPGDSMN1; SMN2ALOX15
SCHEMBL58495 0.89 TUBB1 (0.41) TUBB1GAAHPGDSMN1; SMN2MAPT
SCHEMBL10175741 0.89 TUBB1 (0.45) TUBB1GAAHPGDSMN1; SMN2ALOX15
SCHEMBL12201939 0.89 TUBB1 (0.41) TUBB1GAAHPGDSMN1; SMN2MAPT
SCHEMBL58036 0.89 TUBB1 (0.45) TUBB1GAAHPGDSMN1; SMN2ALOX15
SCHEMBL15429790 0.87 TUBB1 (0.44) TUBB1HPGD
SCHEMBL58501 0.87 TUBB1 (0.44) TUBB1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2374454-A1 Hemiasterlin derivatives and uses thereof in the treatment of cancer Eisai R&D Management Co., Ltd. (JP) 2011-10-12 EP disclosed