SCHEMBL8850690

SCHEMBL8850690

COC(c1ccccc1)c1cccc(Br)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.66
TDO2 P48775 4/20 0.66
ALDH1A1 P00352 4/20 0.41
L3MBTL1 Q9Y468 1/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
CHRM2 P08172 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
CHRM1 P11229 1/20 0.39
DRD1 P21728 1/20 0.39
TBXA2R P21731 1/20 0.39
OPRM1 P35372 1/20 0.39
DRD3 P35462 1/20 0.39
SLC6A3 Q01959 1/20 0.39
MAPK1 P28482 1/20 0.39
LMNA P02545 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28008631 0.86 IDO1 (0.50) IDO1TDO2ALDH1A1L3MBTL1SLC6A2
SCHEMBL73865 0.84 IDO1 (0.70) IDO1TDO2ALDH1A1SLC6A2SLC6A4
SCHEMBL11076842 0.84 IDO1 (0.47) IDO1TDO2ALDH1A1SLC6A2SLC6A4
SCHEMBL9934266 0.82 IDO1 (0.46) IDO1TDO2SLC6A2SLC6A4SLC6A3
SCHEMBL1773224 0.82 SLC6A4 (0.54) IDO1TDO2ALDH1A1L3MBTL1SLC6A2
SCHEMBL461448 0.81 IDO1 (0.47) IDO1TDO2SLC6A2SLC6A4CHRM2
SCHEMBL8851108 0.80 IDO1 (0.60) IDO1TDO2ALDH1A1SLC6A2SLC6A4
SCHEMBL23296602 0.79 IDO1 (0.46) IDO1TDO2SLC6A2SLC6A4CHRM2
SCHEMBL30608097 0.78 IDO1 (0.47) IDO1TDO2ALDH1A1L3MBTL1SLC6A2
SCHEMBL511201 0.78 IDO1 (0.47) IDO1TDO2ALDH1A1L3MBTL1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529444-B1 2-Arylpropenic acids and their utilisation in the preparation of 5-ketoprofen BAYER AG (DE) 1997-04-16 EP disclosed
US-5362907-A Intermediates and their use in the preparation of s-ketoprofen BAYER AKTIENGESELLSCHAFT (DE) 1994-11-08 US disclosed
EP-0529444-A2 2-Arylpropenic acids and their utilisation in the preparation of 5-ketoprofen BAYER AG (DE) 1993-03-03 EP disclosed