SCHEMBL8856483

SCHEMBL8856483

COc1ccc(C(=O)N(N)C2(O)C(=O)c3ccccc3C2=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.50
KMT2A Q03164 2/20 0.50
MAPT P10636 2/20 0.50
RAB9A P51151 2/20 0.50
MAPK1 P28482 1/20 0.50
HPGD P15428 2/20 0.48
KDM4E B2RXH2 1/20 0.48
CES2 O00748 2/20 0.44
CES1 P23141 2/20 0.44
GAA P10253 3/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
OPRM1 P35372 1/20 0.43
OPRL1 P41146 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CA1 P00915 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8856719 0.87 CA1 (0.54) NPC1KMT2AMAPTRAB9AMAPK1
SCHEMBL8856834 0.85 PARP1 (0.49) NPC1KMT2AMAPTRAB9AMAPK1
SCHEMBL8856518 0.84 MAPT (0.46) NPC1KMT2AMAPTRAB9AMAPK1
SCHEMBL8856540 0.84 MAPT (0.47) NPC1KMT2AMAPTRAB9AMAPK1
SCHEMBL8856703 0.83 HCRTR1 (0.46) NPC1KMT2AMAPTRAB9AMAPK1
SCHEMBL8856687 0.82 ALDH1A1 (0.40) NPC1KMT2AMAPTRAB9AMAPK1
SCHEMBL8856566 0.81 CYP1A2 (0.50) KMT2AMAPTRAB9AMAPK1HPGD
SCHEMBL8856578 0.81 CA1 (0.52) NPC1KMT2AMAPTRAB9AMAPK1
SCHEMBL8856819 0.80 CA1 (0.55) NPC1MAPTHPGDKDM4EGAA
SCHEMBL8856498 0.75 HPGD (0.47) KMT2AMAPTHPGDKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5648381-A Derivatives of indan-1,3-dione and indan-1,2,3-trione, methods of preparing them and therapeutic use thereof INNOTHERA (FR) 1997-07-15 US disclosed
EP-0566446-B1 Derivatives of indane-1,3-dione and indane-1,2,3-trione, processes for their preparation and their application in therapy INNOTHERA LAB SA (FR) 1996-02-07 EP disclosed
EP-0566446-A1 Derivatives of indane-1,3-dione and indane-1,2,3-trione, processes for their preparation and their application in therapy INNOTHERA (FR) 1993-10-20 EP disclosed
WO-1993020046-A1 INDAN-1,3-DIONE AND INDAN-1,2,3-TRIONE DERIVATIVES, PROCESSES FOR PREPARATION OF SAME AND THEIR USE AS THERAPEUTIC AGENTS INNOTHERA (FR) 1993-10-14 WO disclosed