SCHEMBL8856580

SCHEMBL8856580

COc1cc2c(=O)c(=O)c(=O)c2cc1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.47
HDAC6 Q9UBN7 1/20 0.45
PTPN1 P18031 1/20 0.45
PPARG P37231 1/20 0.45
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
AKR1B1 P15121 2/20 0.44
CA7 P43166 2/20 0.44
MCL1 Q07820 2/20 0.44
CA9 Q16790 2/20 0.44
CA13 Q8N1Q1 2/20 0.44
RAB9A P51151 2/20 0.44
KLK7 P49862 1/20 0.44
TUBB4A P04350 1/20 0.44
TUBB P07437 1/20 0.44
TUBA3C P0DPH7 1/20 0.44
TUBA1B P68363 1/20 0.44
TUBA4A P68366 1/20 0.44
TUBB4B P68371 1/20 0.44
TUBB3 Q13509 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL9036576 0.98 PTGS2 (0.46) PTGS2HDAC6PTPN1PPARGCA12
SCHEMBL17133045 0.84 MAOB (0.52) PTGS2CA12CA1AKR1B1CA7
SCHEMBL8840801 0.84 MAOB (0.52) PTGS2CA12CA1AKR1B1CA7
SCHEMBL4094512 0.84 MEN1 (0.47) CA1CA7CA9ALDH1A1KDM4E
SCHEMBL8840816 0.81 MAOB (0.50) PTGS2CA12CA1AKR1B1CA7
SCHEMBL17546677 0.81 MAOB (0.50) PTGS2CA12CA1AKR1B1CA7
SCHEMBL8840857 0.81 MAOB (0.50) PTGS2CA12CA1AKR1B1CA7
Water SCHEMBL9036802 0.81 MEN1 (0.46) CA1CA7CA9ALDH1A1KDM4E
SCHEMBL18963272 0.76 MAOB (0.45) MCL1RAB9ATUBB1MAOBALDH1A1
SCHEMBL69624 0.75 MAOB (0.59) CA12CA1AKR1B1CA7MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5648381-A Derivatives of indan-1,3-dione and indan-1,2,3-trione, methods of preparing them and therapeutic use thereof INNOTHERA (FR) 1997-07-15 US disclosed
US-5571843-A Derivatives of indan-1,3-dione and indan-1,2,3-trione, methods of preparing them and therapeutic use thereof INNOTHERA (FR) 1996-11-05 US disclosed
EP-0566446-B1 Derivatives of indane-1,3-dione and indane-1,2,3-trione, processes for their preparation and their application in therapy INNOTHERA LAB SA (FR) 1996-02-07 EP disclosed
EP-0566445-B1 Derivatives of indane 1,3-dione and indane-1,2,3-trione, processes for their preparation and their application in therapy INNOTHERA LAB SA (FR) 1996-02-07 EP disclosed
EP-0566445-A1 Derivatives of indane 1,3-dione and indane-1,2,3-trione, processes for their preparation and their application in therapy INNOTHERA (FR) 1993-10-20 EP disclosed
EP-0566446-A1 Derivatives of indane-1,3-dione and indane-1,2,3-trione, processes for their preparation and their application in therapy INNOTHERA (FR) 1993-10-20 EP disclosed
WO-1993020045-A1 INDAN-1,3-DIONE AND INDAN-1,2,3-TRIONE DERIVATIVES, PROCESSES FOR THE PREPARATION OF SAME AND THEIR APPLICATION AS THERAPEUTIC AGENTS INNOTHERA (FR) 1993-10-14 WO disclosed
WO-1993020046-A1 INDAN-1,3-DIONE AND INDAN-1,2,3-TRIONE DERIVATIVES, PROCESSES FOR PREPARATION OF SAME AND THEIR USE AS THERAPEUTIC AGENTS INNOTHERA (FR) 1993-10-14 WO disclosed