SCHEMBL8856855

SCHEMBL8856855

COC(=O)N(N)C1(O)C(=O)c2ccc(OC)cc2C1=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.59
CA2 P00918 2/20 0.59
CA7 P43166 2/20 0.59
CA9 Q16790 2/20 0.59
CA4 P22748 1/20 0.59
KMT2A Q03164 6/20 0.41
MEN1 O00255 5/20 0.41
GAA P10253 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPT P10636 3/20 0.36
RAB9A P51151 3/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8856719 0.82 CA1 (0.54) CA1CA2CA7CA9CA4
SCHEMBL8856578 0.81 CA1 (0.52) CA1CA2CA7CA9CA4
SCHEMBL8856819 0.80 CA1 (0.55) CA1CA2CA7CA9CA4
SCHEMBL11137560 0.75 CA1 (0.79) CA1CA2CA7CA9CA4
SCHEMBL4395035 0.75 CA1 (1.00) CA1CA2CA7CA9CA4
Water SCHEMBL1222259 0.74 CA1 (0.96) CA1CA2CA7CA9CA4
SCHEMBL8856483 0.72 NPC1 (0.50) CA1CA2CA7CA9CA4
SCHEMBL8856834 0.72 PARP1 (0.49) CA1CA2CA7CA9CA4
SCHEMBL8856863 0.70 CA1 (0.60) CA1CA2CA7CA9CA4
SCHEMBL8856679 0.68 CA1 (0.56) CA1CA2CA7CA9CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5648381-A Derivatives of indan-1,3-dione and indan-1,2,3-trione, methods of preparing them and therapeutic use thereof INNOTHERA (FR) 1997-07-15 US disclosed
EP-0566446-B1 Derivatives of indane-1,3-dione and indane-1,2,3-trione, processes for their preparation and their application in therapy INNOTHERA LAB SA (FR) 1996-02-07 EP disclosed
EP-0566446-A1 Derivatives of indane-1,3-dione and indane-1,2,3-trione, processes for their preparation and their application in therapy INNOTHERA (FR) 1993-10-20 EP disclosed
WO-1993020046-A1 INDAN-1,3-DIONE AND INDAN-1,2,3-TRIONE DERIVATIVES, PROCESSES FOR PREPARATION OF SAME AND THEIR USE AS THERAPEUTIC AGENTS INNOTHERA (FR) 1993-10-14 WO disclosed