SCHEMBL8864740

SCHEMBL8864740

O=C(O)c1ccccc1C(=O)c1ccncc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.73
MEN1 O00255 2/20 0.67
KMT2A Q03164 2/20 0.67
CDC25B P30305 2/20 0.63
ATM Q13315 1/20 0.63
NR4A1 P22736 1/20 0.61
CDC25A P30304 1/20 0.58
HSD17B10 Q99714 1/20 0.58
ALDH1A1 P00352 4/20 0.56
ALOX15 P16050 2/20 0.56
NAPRT Q6XQN6 1/20 0.56
KDM4E B2RXH2 1/20 0.52
POLB P06746 2/20 0.51
PLOD2 O00469 1/20 0.50
PLOD3 O60568 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
HPGD P15428 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
2-Benzoylbenzoic Acid SCHEMBL76332 0.85 AKR1C3 (1.00) AKR1C3CDC25BATMNR4A1CDC25A
2-Benzoylbenzoic Acid SCHEMBL30296847 0.85 AKR1C3 (1.00) AKR1C3CDC25BATMNR4A1CDC25A
SCHEMBL27524893 0.85 AKR1C3 (0.91) AKR1C3CDC25BATMNR4A1CDC25A
2-Benzoylbenzoic Acid SCHEMBL1525895 0.83 AKR1C3 (0.95) AKR1C3CDC25BATMNR4A1CDC25A
2-Benzoylbenzoic Acid SCHEMBL10979285 0.83 AKR1C3 (0.95) AKR1C3CDC25BATMNR4A1CDC25A
2-Benzoylbenzoic Acid SCHEMBL9317427 0.83 AKR1C3 (0.95) AKR1C3CDC25BATMNR4A1CDC25A
2-Benzoylbenzoic Acid SCHEMBL11577549 0.83 AKR1C3 (0.95) AKR1C3CDC25BATMNR4A1CDC25A
2-Benzoylbenzoic Acid SCHEMBL3791911 0.83 AKR1C3 (0.95) AKR1C3CDC25BATMNR4A1CDC25A
2-Benzoylbenzoic Acid SCHEMBL9562236 0.83 AKR1C3 (0.95) AKR1C3CDC25BATMNR4A1CDC25A
2-Benzoylbenzoic Acid SCHEMBL7768301 0.83 AKR1C3 (0.95) AKR1C3CDC25BATMNR4A1CDC25A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9638690-B2 Compounds and compositions for use as alkylating agent sensors and methods of use thereof THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2017-05-02 US disclosed
US-9638690-B2 Compounds and compositions for use as alkylating agent sensors and methods of use thereof THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2017-05-02 US disclosed
US-20160131641-A1 COMPOUNDS AND COMPOSITIONS FOR USE AS ALKYLATING AGENT SENSORS AND METHODS OF USE THEREOF THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2016-05-12 US disclosed
US-20160131641-A1 COMPOUNDS AND COMPOSITIONS FOR USE AS ALKYLATING AGENT SENSORS AND METHODS OF USE THEREOF THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2016-05-12 US disclosed
US-5624922-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1997-04-29 US disclosed
EP-0597540-B1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC (US) 1996-06-05 EP disclosed
US-5380721-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1995-01-10 US disclosed
EP-0597540-A1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1994-05-18 EP disclosed
US-5268372-A Where nitrogen in position 2 and 5 are connected by a methylene bridge STERLING WINTHROP INC. (US) 1993-12-07 US disclosed
US-5206231-A 2,5-benzodiazocine antiarrhythmic agents STERLING DRUG INC. (US) 1993-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160131641-A1 COMPOUNDS AND COMPOSITIONS FOR USE AS ALKYLATING AGENT SENSORS AND METHODS OF USE THEREOF MGMT, MCL1, OGG1 AKR1C3 3472/4885MEN1 341/4885KMT2A 311/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.