SCHEMBL8864801

SCHEMBL8864801

C/C(=C\c1ccc(Oc2ccccc2)cc1)C(=O)O

nearest known ligand 0.69

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.69
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
ALDH1A1 P00352 2/20 0.51
MEN1 O00255 1/20 0.51
LMNA P02545 1/20 0.51
KMT2A Q03164 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
SMN1; SMN2 Q16637 3/20 0.49
SRD5A2 P31213 2/20 0.47
ESR1 P03372 1/20 0.47
PARP10 Q53GL7 1/20 0.46
HTT P42858 2/20 0.45
HPGD P15428 1/20 0.45
TBXAS1 P24557 2/20 0.44
RECQL P46063 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8864809 1.00 AKR1C3 (0.69) AKR1C3NPC1RAB9AALDH1A1MEN1
SCHEMBL10987986 0.85 TBXAS1 (0.59) AKR1C3NPC1RAB9AALDH1A1LMNA
SCHEMBL10987989 0.85 TBXAS1 (0.59) AKR1C3NPC1RAB9AALDH1A1LMNA
SCHEMBL21470276 0.85 AKR1C3 (0.62) AKR1C3NPC1RAB9AALDH1A1MEN1
Hydrochloric Acid SCHEMBL10992507 0.84 TBXAS1 (0.61) AKR1C3NPC1RAB9AALDH1A1LMNA
Hydrochloric Acid SCHEMBL10982425 0.84 TBXAS1 (0.61) AKR1C3NPC1RAB9AALDH1A1LMNA
SCHEMBL37034 0.82 AKR1C3 (1.00) AKR1C3NPC1RAB9AALDH1A1MEN1
SCHEMBL581982 0.82 AKR1C3 (1.00) AKR1C3NPC1RAB9AALDH1A1MEN1
SCHEMBL41906 0.82 AKR1C3 (1.00) AKR1C3NPC1RAB9AALDH1A1MEN1
SCHEMBL16568719 0.82 AKR1C3 (1.00) AKR1C3NPC1RAB9AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019196714-A1 N-SUBSTITUTED ACRYLAMIDE DERIVATIVE AS DHODH INHIBITOR, AND PREPARATION AND USE THEREOF 华东理工大学 2019-10-17 WO disclosed
US-5646313-A PREPARING ENKEPHALINASE INHIBITORS SOCIETE CIVILE BIOPROJET (FR) 1997-07-08 US disclosed
US-5612371-A ENZYME INHIBITORS SOCIETE CIVILE BIOPROJECT (FR) 1997-03-18 US disclosed
EP-0009683-A1 Basic phenyl ethers, pharmaceutical compositions containing them and the preparation of these ethers and compositions MERCK PATENT GmbH (DE) 1980-04-16 EP disclosed