SCHEMBL8865503

SCHEMBL8865503

CCOc1ccc(/C=C(\CBr)C(=O)O)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HTT P42858 1/20 0.48
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48
RELA Q04206 1/20 0.47
MAOB P27338 6/20 0.46
MAOA P21397 1/20 0.44
ALOX5 P09917 1/20 0.44
NR1H4 Q96RI1 1/20 0.44
NQO1 P15559 1/20 0.44
PARP10 Q53GL7 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.43
PLA2G4B P0C869 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865510 1.00 NPC1 (0.48) NPC1RAB9AKDM4EALDH1A1HTT
SCHEMBL8864815 0.88 ALOX5 (0.51) NPC1RAB9AKDM4EALDH1A1KMT2A
SCHEMBL8864827 0.88 ALOX5 (0.51) NPC1RAB9AKDM4EALDH1A1KMT2A
SCHEMBL8865614 0.84 GSK3B (0.50) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL8865604 0.84 GSK3B (0.50) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL8415544 0.82 AKR1C3 (0.56) NPC1RAB9AKDM4EALDH1A1HTT
SCHEMBL4579188 0.82 AKR1C3 (0.56) NPC1RAB9AKDM4EALDH1A1HTT
SCHEMBL11250951 0.80 NR1H4 (0.55) NPC1RAB9AKDM4EALDH1A1HTT
SCHEMBL8865036 0.80 MAPT (0.44) NPC1RAB9AKDM4EALDH1A1HTT
SCHEMBL8865053 0.80 MAPT (0.44) NPC1RAB9AKDM4EALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5646313-A PREPARING ENKEPHALINASE INHIBITORS SOCIETE CIVILE BIOPROJET (FR) 1997-07-08 US disclosed
US-5612371-A ENZYME INHIBITORS SOCIETE CIVILE BIOPROJECT (FR) 1997-03-18 US disclosed