SCHEMBL8865663

SCHEMBL8865663

N#Cc1ccc2nc(-c3ccc(C(=O)O)cc3)cn2c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.62
ALDH1A3 P47895 7/20 0.61
ALDH1A1 P00352 11/20 0.56
KDM4E B2RXH2 8/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
HSP90AA1 P07900 1/20 0.56
RXFP1 Q9HBX9 1/20 0.56
NPC1 O15118 8/20 0.48
RAB9A P51151 8/20 0.48
SMN1; SMN2 Q16637 5/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
POLB P06746 3/20 0.47
GAA P10253 2/20 0.47
ALDH1A2 O94788 1/20 0.47
GLA P06280 1/20 0.44
MITF O75030 1/20 0.44
KDM5A P29375 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8867230 0.99 APP (0.61) APPALDH1A3ALDH1A1KDM4EMEN1
SCHEMBL2127570 0.92 ALDH1A3 (0.65) APPALDH1A3ALDH1A1KDM4EMEN1
Bromide SCHEMBL8866701 0.91 ALDH1A3 (0.64) APPALDH1A3ALDH1A1KDM4EMEN1
SCHEMBL4952001 0.84 ALDH1A3 (0.78) APPALDH1A3ALDH1A1KDM4EMEN1
SCHEMBL5301325 0.83 ALDH1A3 (0.86) APPALDH1A3ALDH1A1KDM4EMEN1
SCHEMBL14046613 0.83 ALDH1A3 (0.81) APPALDH1A3ALDH1A1KDM4EMEN1
SCHEMBL8866225 0.82 ALDH1A3 (0.49) APPALDH1A3ALDH1A1KDM4EMEN1
SCHEMBL2128252 0.81 APP (0.74) APPALDH1A3ALDH1A1KDM4EMEN1
Bromide SCHEMBL8867379 0.81 ALDH1A3 (0.48) APPALDH1A3ALDH1A1KDM4EMEN1
SCHEMBL4952240 0.80 APP (0.68) APPALDH1A3ALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614531-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-03-25 US disclosed
EP-0668278-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1995-08-23 EP disclosed