SCHEMBL8865751

SCHEMBL8865751

CCOC(=O)Cc1ccc(C#Cc2ccc3c(c2)C(C)(C)CC(C)(C)O3)nc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.49
RARA P10276 1/20 0.49
RARB P10826 1/20 0.49
RARG P13631 1/20 0.49
KMT2A Q03164 1/20 0.49
ACACB O00763 4/20 0.38
CYP26A1 O43174 2/20 0.38
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
CASP1 P29466 1/20 0.36
HSD17B10 Q99714 1/20 0.36
FDFT1 P37268 1/20 0.35
SSTR5 P35346 1/20 0.34
JAK2 O60674 2/20 0.34
JAK1 P23458 2/20 0.34
TYK2 P29597 2/20 0.34
JAK3 P52333 2/20 0.34
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9209527 0.91 CYP3A4 (0.47) CYP3A4RARARARBRARGKMT2A
SCHEMBL8865044 0.89 CYP3A4 (0.46) CYP3A4RARARARBRARGKMT2A
SCHEMBL8876189 0.88 CYP26A1 (0.43) CYP3A4RARARARBRARGKMT2A
SCHEMBL8865372 0.87 CYP3A4 (0.45) CYP3A4RARARARBRARGKMT2A
SCHEMBL8865618 0.86 CYP3A4 (0.39) CYP3A4RARARARBRARGKMT2A
SCHEMBL9866199 0.86 CYP3A4 (0.44) CYP3A4RARARARBRARGKMT2A
SCHEMBL8626930 0.86 CYP3A4 (0.65) CYP3A4RARARARBRARGKMT2A
SCHEMBL8864919 0.86 CYP3A4 (0.38) CYP3A4RARARARBRARGKMT2A
SCHEMBL8865446 0.85 CYP3A4 (0.43) CYP3A4RARARARBRARGKMT2A
SCHEMBL8865454 0.84 CYP3A4 (0.43) CYP3A4RARARARBRARGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5677323-A SKIN DISORDERS, PSORIASIS ALLERGAN (US) 1997-10-14 US disclosed