SCHEMBL8866907

SCHEMBL8866907

NCC(=O)NC(Cc1ccccc1)c1ccc(OC(=O)/C=C\C(=O)Oc2ccc(C(Cc3ccccc3)NC(=O)CN)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
HTT P42858 1/20 0.52
NCOA1 Q15788 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
NCOA3 Q9Y6Q9 1/20 0.52
CTSC P53634 2/20 0.47
MMP2 P08253 1/20 0.43
SOAT1 P35610 1/20 0.42
CNR2 P34972 2/20 0.41
CCR3 P51677 1/20 0.41
LTA4H P09960 1/20 0.41
FAAH O00519 1/20 0.41
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9054827 0.85 CNR2 (0.58) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
SCHEMBL6813188 0.84 ALDH1A1 (0.71) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
SCHEMBL16889096 0.84 ALDH1A1 (0.71) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
SCHEMBL8866666 0.82 ALDH1A1 (0.52) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
Hydrochloric Acid SCHEMBL6813768 0.82 ALDH1A1 (0.69) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
SCHEMBL5304987 0.81 ALDH1A1 (0.60) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
Fumaric Acid SCHEMBL8866914 0.81 ALDH1A1 (0.53) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
Maleic Acid SCHEMBL8866899 0.81 ALDH1A1 (0.53) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
SCHEMBL9054159 0.80 ALDH1A1 (0.55) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3
SCHEMBL9322630 0.78 ALDH1A1 (0.58) ALDH1A1HTTNCOA1SMN1; SMN2NCOA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605916-A Arylalkyl-amines having anticonvulsant and neuroprotective properties ASTRA AB (SE) 1997-02-25 US disclosed
US-5539120-A Arylalkyl-amines having anticonvulsant and neuroprotective properties AGENCE SPATIALE EUROPEENNE (FR) 1996-07-23 US disclosed
EP-0356035-B1 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties ASTRA AB (SE) 1996-03-13 EP disclosed
US-5430044-A Arylalkyl-amines and -amides having anticonvulsant and neuroprotective properties FISONS CORPORATION (GB) 1995-07-04 US disclosed
EP-0648489-A1 Arylalkylamides having neuroprotective properties FISONS CORPORATION (US) 1995-04-19 EP disclosed
EP-0648745-A1 Arylalkylamine having anticonvulsant and neuroprotective properties Astra Aktiebolag (SE) 1995-04-19 EP disclosed
US-5331007-A Arylalkyl-amines and -amides having anticonvulsant and neuroprotective properties FISONS CORPORATION (US) 1994-07-19 US disclosed
WO-1991011995-A1 ARYLALKYL-AMINES AND -AMIDES HAVING ANTICONVULSANT AND NEUROPROTECTIVE PROPERTIES FISONS CORPORATION (US) 1991-08-22 WO disclosed