SCHEMBL8868630

SCHEMBL8868630

S=C=Nc1ccc(Nc2ccncc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 1/20 0.48
P2RY6 Q15077 2/20 0.44
MIF P14174 1/20 0.43
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CTSD P07339 1/20 0.38
POLB P06746 2/20 0.36
MAPT P10636 2/20 0.36
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
HSD17B10 Q99714 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1848797 0.88 MIF (0.54) P2RY6MIFCA1CA2MAPT
SCHEMBL5572886 0.81
SCHEMBL11699033 0.80 MIF (0.64) P2RY6MIFCA1CA2POLB
SCHEMBL11697691 0.78 HPGD (0.48) P2RY6MIFCA1CA2MAPT
SCHEMBL11696524 0.78 P2RY6 (0.45) P2RY6MIFCA1CA2POLB
SCHEMBL5725177 0.78 P2RY6 (0.48) P2RY6MIFCA1CA2MAPT
SCHEMBL11693832 0.76 CYP1B1 (0.49) P2RY6MIFCA1CA2POLB
SCHEMBL1333233 0.74 P2RY6 (0.45) P2RY6MIFCA1CA2HSD17B10
Bitoscanate SCHEMBL157128 0.73 MIF (0.72) P2RY6MIFCA1CA2MAPT
SCHEMBL725063 0.73 RAD52 (0.70) RAD52CTSDPOLBMAPTADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5665746-A BACTERICIDE HOFFMANN-LA ROCHE INC. (US) 1997-09-09 US disclosed
US-5594135-A BACTERICIDES HOFFMANN-LA ROCHE INC. (US) 1997-01-14 US disclosed
US-5589473-A BACTERICIDES HOFFMANN-LA ROCHE INC. (US) 1996-12-31 US disclosed
EP-0675122-A2 Mono or bicyclic DNA gyrase inhibitors F. HOFFMANN-LA ROCHE AG (CH) 1995-10-04 EP disclosed