SCHEMBL8869907

SCHEMBL8869907

[CH2]c1ccccc1-n1cnc2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.56
POLB P06746 1/20 0.51
FGFR1 P11362 3/20 0.50
MKNK1 Q9BUB5 1/20 0.49
MKNK2 Q9HBH9 1/20 0.49
ALDH1A1 P00352 1/20 0.46
ROCK1 Q13464 1/20 0.45
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3417306 0.86 HTT (0.73) HTTPOLBFGFR1MKNK1MKNK2
SCHEMBL23266636 0.81 HTT (0.60) HTTPOLBFGFR1MKNK1MKNK2
SCHEMBL56852 0.79 FGFR1 (0.61) HTTPOLBFGFR1ALDH1A1
SCHEMBL23840256 0.79 HTT (0.58) HTTPOLBFGFR1MKNK1MKNK2
SCHEMBL4944401 0.78 HTT (0.56) HTTPOLBFGFR1MKNK1MKNK2
SCHEMBL23840275 0.78 FGFR1 (0.58) HTTPOLBFGFR1MKNK1MKNK2
SCHEMBL5937 0.78 HTT (0.56) HTTPOLBFGFR1MKNK1MKNK2
SCHEMBL8624088 0.78 FGFR1 (0.59) HTTPOLBFGFR1ALDH1A1
SCHEMBL7211112 0.78 HTT (0.56) HTTPOLBFGFR1ALDH1A1ROCK1
SCHEMBL12138417 0.78 HTT (0.56) HTTPOLBFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991644-A2 NONSTEROIDAL AND STEROIDAL COMPOUNDS WITH POTENT ANDROGEN RECEPTOR DOWN-REGULATION AND ANTI PROSTATE CANCER ACTIVITY University of Maryland, Baltimore (US) 2016-03-09 EP disclosed
WO-2014165815-A2 NONSTEROIDAL AND STEROIDAL COMPOUNDS WITH POTENT ANDROGEN RECEPTOR DOWN-REGULATION AND ANTI PROSTATE CANCER ACTIVITY UNIVERSITY OF MARYLAND, BALTIMORE (US) 2014-10-09 WO disclosed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US disclosed