SCHEMBL8870075

SCHEMBL8870075

COc1ccc(Oc2ccc3[nH]c(C(=O)O)cc3c2)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.78
XDH P47989 1/20 0.67
PDGFRB P09619 2/20 0.66
PDGFRA P16234 2/20 0.66
FLT3 P36888 6/20 0.60
CYP1A2 P05177 2/20 0.60
CYP2C9 P11712 2/20 0.60
MEN1 O00255 1/20 0.60
CYP3A4 P08684 1/20 0.60
TSHR P16473 1/20 0.60
HDAC6 Q9UBN7 1/20 0.60
KDM4E B2RXH2 3/20 0.57
ALDH1A1 P00352 3/20 0.57
HPGD P15428 2/20 0.57
NPC1 O15118 1/20 0.57
LMNA P02545 1/20 0.57
HTT P42858 1/20 0.57
RAB9A P51151 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
PIN1 Q13526 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL335235 0.91 PDGFRB (0.79) KMT2APDGFRBPDGFRAFLT3CYP1A2
SCHEMBL8869244 0.88 KMT2A (0.78) KMT2AXDHPDGFRBPDGFRAFLT3
SCHEMBL9513175 0.88 KMT2A (1.00) KMT2AXDHPDGFRBPDGFRAFLT3
SCHEMBL31287858 0.85 KMT2A (0.78) KMT2AXDHPDGFRBPDGFRAFLT3
SCHEMBL9816551 0.85 KMT2A (0.78) KMT2AXDHPDGFRBPDGFRAFLT3
SCHEMBL4263996 0.85 PDGFRB (0.61) KMT2APDGFRBPDGFRAFLT3CYP1A2
SCHEMBL8868735 0.82 RAB9A (0.85) KMT2AXDHPDGFRBPDGFRAFLT3
SCHEMBL31287830 0.82 KMT2A (0.72) KMT2AXDHPDGFRBPDGFRAFLT3
SCHEMBL31287750 0.81 KMT2A (0.72) KMT2AXDHFLT3CYP1A2CYP2C9
SCHEMBL6866887 0.80 PDGFRB (1.00) KMT2APDGFRBPDGFRAFLT3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637593-A MIGRAINE; HYPOTENSIVE AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-06-10 US disclosed