SCHEMBL8870530

SCHEMBL8870530

OC(c1ccc(Br)cc1)(c1ccc(Br)cc1)c1cncnc1

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 17/20 0.66
CYP3A4 P08684 1/20 0.53
CYP3A5 P20815 1/20 0.53
USP2 O75604 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8870773 0.87 CYP3A4 (0.52) CYP19A1CYP3A4CYP3A5
SCHEMBL31124841 0.82 CYP2A6 (0.50) CYP19A1USP2RAB9A
SCHEMBL9651054 0.79 CYP19A1 (1.00) CYP19A1CYP3A4CYP3A5
SCHEMBL913343 0.78 CYP19A1 (0.79) CYP19A1CYP3A4CYP3A5
SCHEMBL17159521 0.77 CYP19A1 (0.53) CYP19A1CYP3A4CYP3A5
SCHEMBL8870724 0.75 CYP19A1 (0.59) CYP19A1CYP3A4CYP3A5
SCHEMBL10631898 0.73 CYP19A1 (0.86) CYP19A1CYP3A4CYP3A5USP2RAB9A
SCHEMBL27282169 0.73 CYP19A1 (0.86) CYP19A1CYP3A4CYP3A5
SCHEMBL4432529 0.73 ALDH1A1 (0.48) CYP19A1CYP3A4
SCHEMBL13865450 0.73 ALDH1A1 (0.48) CYP19A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637605-A ANTITUMOR AGENTS CIBA GEIGY CORPORATION (US) 1997-06-10 US disclosed
US-5583128-A ADMINISTERING A SIDE EFFECT REDUCED AROMATASE INHIBITOR CIBA-GEIGY CORPORATION (US) 1996-12-10 US disclosed
US-5457209-A Antitumor agents CIBA-GEIGY CORPORATION (US) 1995-10-10 US disclosed
US-5376669-A Antitumor agents CIBA-GEIGY CORP. (US) 1994-12-27 US disclosed
US-5227393-A estrogen-dependent diseases, anticancer CIBA-GEIGY CORPORATION (US) 1993-07-13 US disclosed
EP-0490816-A2 Fluoro-compounds CIBA-GEIGY AG (CH) 1992-06-17 EP disclosed