SCHEMBL8870947

SCHEMBL8870947

CCc1cc(C#N)ccc1Nc1c(NC(C)c2ccccc2)c(=O)c1=O

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.72
ABCC8 Q09428 1/20 0.72
KCNJ11 Q14654 1/20 0.72
KCNJ8 Q15842 1/20 0.72
CXCR2 P25025 6/20 0.48
MAPKAPK2 P49137 9/20 0.47
AURKB Q96GD4 3/20 0.47
ROCK1 Q13464 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47
PDGFRA P16234 2/20 0.47
MAPK1 P28482 2/20 0.47
CSNK1G1 Q9HCP0 2/20 0.47
DCLK1 O15075 1/20 0.47
ROCK2 O75116 1/20 0.47
CHEK2 O96017 1/20 0.47
GSK3A P49840 1/20 0.47
GSK3B P49841 1/20 0.47
IRAK1 P51617 1/20 0.47
PRKX P51817 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8870945 1.00 ABCC9 (0.72) ABCC9ABCC8KCNJ11KCNJ8CXCR2
SCHEMBL8870610 0.86 ABCC9 (0.53) ABCC9ABCC8KCNJ11KCNJ8CXCR2
SCHEMBL8870608 0.86 ABCC9 (0.53) ABCC9ABCC8KCNJ11KCNJ8CXCR2
SCHEMBL6024203 0.84 ABCC9 (1.00) ABCC9ABCC8KCNJ11KCNJ8CXCR2
SCHEMBL4258934 0.84 ABCC9 (1.00) ABCC9ABCC8KCNJ11KCNJ8CXCR2
SCHEMBL8870870 0.79 MAPKAPK2 (0.65) CXCR2MAPKAPK2AURKBROCK1CYP3A4
SCHEMBL9146091 0.79 MAPKAPK2 (0.65) CXCR2MAPKAPK2AURKBROCK1CYP3A4
SCHEMBL8871512 0.79 MAPKAPK2 (0.65) CXCR2MAPKAPK2AURKBROCK1CYP3A4
SCHEMBL8868951 0.79 MAPKAPK2 (0.59) CXCR2MAPKAPK2AURKBROCK1CYP3A4
SCHEMBL9148198 0.79 MAPKAPK2 (0.59) CXCR2MAPKAPK2AURKBROCK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5466712-A Smooth muscle relaxants AMERICAN HOME PRODUCTS CORPORATION (US) 1995-11-14 US claimed
US-5605909-A REDUCING ADVERSE EFFECTS OF SMOOTH MUSCLE CONTRACTIONS AMERICAN HOME PRODUCTS CORPORATION (US) 1997-02-25 US disclosed
US-5532245-A TO REDUCE SMOOTH MUSCLE CONTRACTIONS; TREATMENT FOR URINARY INCONTINENCE, IRITABLE BOWEL SYNDROME AMERICAN HOME PRODUCTS CORPORATION (US) 1996-07-02 US disclosed
US-5466712-A Smooth muscle relaxants AMERICAN HOME PRODUCTS CORPORATION (US) 1995-11-14 US disclosed