SCHEMBL8875508

SCHEMBL8875508

COc1ccccc1N1CCN(CCCNC(=O)c2cccc3c(=O)c(C)c(C(C)(C)C)oc23)CC1

nearest known ligand 0.78

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.78
ADRA1D P25100 4/20 0.78
ADRA1A P35348 4/20 0.78
ADRA1B P35368 4/20 0.78
DRD3 P35462 9/20 0.62
DRD2 P14416 10/20 0.58
FAAH O00519 1/20 0.56
CNR1 P21554 1/20 0.56
DRD4 P21917 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8877020 0.98 HTR1A (0.76) HTR1AADRA1DADRA1AADRA1BDRD3
SCHEMBL8874517 0.93 HTR1A (0.77) HTR1AADRA1DADRA1AADRA1BDRD3
SCHEMBL8877526 0.92 HTR1A (0.75) HTR1AADRA1DADRA1AADRA1BDRD3
SCHEMBL8875092 0.90 HTR1A (0.82) HTR1AADRA1DADRA1AADRA1BDRD3
SCHEMBL8877282 0.90 HTR1A (0.73) HTR1AADRA1DADRA1AADRA1BDRD3
SCHEMBL9567529 0.90 HTR1A (0.73) HTR1AADRA1DADRA1AADRA1BDRD3
Upidosin SCHEMBL6638869 0.88 HTR1A (1.00) HTR1AADRA1DADRA1AADRA1BDRD3
Upidosin SCHEMBL29387625 0.88 HTR1A (1.00) HTR1AADRA1DADRA1AADRA1BDRD3
SCHEMBL8875957 0.87 HTR1A (0.77) HTR1AADRA1DADRA1AADRA1BDRD3
Upidosin SCHEMBL8875378 0.86 HTR1A (0.97) HTR1AADRA1DADRA1AADRA1BDRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605896-A Bicyclic heterocyclic derivatives having α1 adrenergic and 5HT1A activities RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1997-02-25 US claimed
EP-0558245-A1 Heterobicyclic compounds as antagogists of alpha-1 adrenergic and SHT1A receptors RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 1993-09-01 EP claimed