SCHEMBL8875995

SCHEMBL8875995

CC=Cc1cccc2c(=O)c(OCc3ccccc3)c(-c3ccccc3)oc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.45
ABCG2 Q9UNQ0 9/20 0.45
ABCC1 P33527 2/20 0.45
KDM4E B2RXH2 4/20 0.43
GAA P10253 2/20 0.43
KCNA3 P22001 1/20 0.42
HSD17B10 Q99714 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP1A1 P04798 2/20 0.41
CYP1B1 Q16678 2/20 0.41
CYP1A2 P05177 1/20 0.41
ALDH1A1 P00352 3/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8875983 1.00 PPARG (0.45) PPARGABCG2ABCC1KDM4EGAA
SCHEMBL8875978 1.00 PPARG (0.45) PPARGABCG2ABCC1KDM4EGAA
SCHEMBL8876901 0.85 ABCG2 (0.62) ABCG2ABCC1KDM4EGAAHSD17B10
SCHEMBL8876891 0.85 ABCG2 (0.62) ABCG2ABCC1KDM4EGAAHSD17B10
SCHEMBL10801230 0.78 LMNA (0.47) ABCG2ABCC1KDM4EGAAKMT2A
SCHEMBL10801234 0.78 LMNA (0.47) ABCG2ABCC1KDM4EGAAKMT2A
SCHEMBL8876174 0.78 CYSLTR1 (0.52) PPARGABCG2ABCC1KDM4EGAA
SCHEMBL8875292 0.77 ABCG2 (0.58) ABCG2KDM4EGAAHSD17B10KMT2A
SCHEMBL8875308 0.77 ABCG2 (0.58) ABCG2KDM4EGAAHSD17B10KMT2A
SCHEMBL8875296 0.77 ABCG2 (0.58) ABCG2KDM4EGAAHSD17B10KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605896-A Bicyclic heterocyclic derivatives having α1 adrenergic and 5HT1A activities RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1997-02-25 US disclosed
US-5474994-A Treating hypertension, urethral and lower urinary tract contractions RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1995-12-12 US disclosed