SCHEMBL8876451

SCHEMBL8876451

COc1ccccc1N1CCN(CCNC(=O)Nc2cccc3c(=O)c(C)c(-c4ccccc4)oc23)CC1

nearest known ligand 0.78

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.71
ADRA1A P35348 5/20 0.71
ADRA1D P25100 3/20 0.71
ADRA1B P35368 3/20 0.71
LMNA P02545 3/20 0.65
USP2 O75604 1/20 0.65
MAPT P10636 1/20 0.65
KMT2A Q03164 1/20 0.65
ALDH1A1 P00352 1/20 0.62
DRD2 P14416 7/20 0.59
DRD4 P21917 7/20 0.59
DRD3 P35462 7/20 0.59
ADRA2A P08913 2/20 0.59
DRD1 P21728 2/20 0.59
DRD5 P21918 2/20 0.59
HTR2A P28223 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8875111 0.97 HTR1A (0.67) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8876770 0.89 HTR1A (0.68) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8877818 0.89 HTR1A (0.69) HTR1AADRA1AADRA1DADRA1BLMNA
Hydrochloric Acid SCHEMBL8874106 0.88 HTR1A (0.67) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8876462 0.88 HTR1A (0.67) HTR1AADRA1AADRA1DADRA1BLMNA
Hydrochloric Acid SCHEMBL8875648 0.88 HTR1A (0.69) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8875435 0.88 HTR1A (0.71) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8879180 0.87 HTR1A (0.91) HTR1AADRA1AADRA1DADRA1BLMNA
Hydrochloric Acid SCHEMBL8875518 0.86 HTR1A (0.88) HTR1AADRA1AADRA1DADRA1BLMNA
Hydrochloric Acid SCHEMBL8875523 0.86 HTR1A (0.88) HTR1AADRA1AADRA1DADRA1BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605896-A Bicyclic heterocyclic derivatives having α1 adrenergic and 5HT1A activities RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1997-02-25 US claimed
US-5403842-A Adrenergic blocking and antiserotonine agents; urogenital disorders including spasms of the urethral tract and prostrate problems RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1995-04-04 US claimed
EP-0558245-A1 Heterobicyclic compounds as antagogists of alpha-1 adrenergic and SHT1A receptors RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 1993-09-01 EP claimed