SCHEMBL8876589

SCHEMBL8876589

Cc1c(-c2ccccc2)nc(C2CC2)c(C=O)c1-c1ccc(F)cc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PRKAA2 P54646 1/20 0.46
RXRA P19793 2/20 0.45
NR1I2 O75469 1/20 0.41
NR4A2 P43354 1/20 0.41
PDE4D Q08499 1/20 0.41
HMGCR P04035 1/20 0.39
AR P10275 1/20 0.39
PTGS2 P35354 1/20 0.39
DHODH Q02127 3/20 0.38
PLAT P00750 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8878297 0.86 RXRA (0.48) PRKAA2RXRANR1I2NR4A2PDE4D
SCHEMBL8878292 0.86 RXRA (0.48) PRKAA2RXRANR1I2NR4A2PDE4D
SCHEMBL8876604 0.85 PRKAA2 (0.46) PRKAA2RXRANR1I2NR4A2PDE4D
SCHEMBL8878327 0.81 DHODH (0.51) PRKAA2RXRADHODH
SCHEMBL8878051 0.81 PRKAA2 (0.66) PRKAA2RXRADHODH
SCHEMBL244423 0.79 RXRA (0.67) PRKAA2RXRANR1I2NR4A2PDE4D
SCHEMBL29419163 0.79 RXRA (0.67) PRKAA2RXRANR1I2NR4A2PDE4D
SCHEMBL8877504 0.79 PRKAA2 (0.46) PRKAA2RXRADHODHALDH1A1
SCHEMBL8876748 0.78 AR (0.42) ARPTGS2DHODHALDH1A1
SCHEMBL8879706 0.78 GCGR (0.44) HMGCRARDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed
US-5506219-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-04-09 US disclosed
EP-0444533-A2 Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1991-09-04 EP disclosed