SCHEMBL8877201

SCHEMBL8877201

CO[PH](=O)C(C#Cc1c(-c2ccc(F)cc2)cc(C2CC2)nc1C(C)C)(C(=O)O)C(C)O

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
HMGCR P04035 1/20 0.37
MAPT P10636 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8878657 0.96 HMGCR (0.42) NPSR1KDM4EHTTL3MBTL1ADORA2A
SCHEMBL8877694 0.91 ADORA2A (0.40) NPSR1KDM4EHTTL3MBTL1ADORA2A
SCHEMBL8877064 0.89 SQOR (0.43) NPSR1KDM4E
SCHEMBL8877354 0.87 HMGCR (0.43) NPSR1KDM4EHTTL3MBTL1ADORA2A
SCHEMBL8877221 0.85
SCHEMBL8878176 0.80 SQOR (0.42) NPSR1KDM4EADORA2AADORA1MAPT
SCHEMBL8901879 0.80 HMGCR (0.36) NPSR1KDM4EHTTL3MBTL1ADORA2A
SCHEMBL8877339 0.80 SQOR (0.40)
SCHEMBL8877271 0.79 GCGR (0.34)
SCHEMBL8878097 0.79 GCGR (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed