SCHEMBL8877460

SCHEMBL8877460

CC(C)(C)OC(=O)N1c2ncccc2CC1O

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.43
GPR119 Q8TDV5 9/20 0.42
GRM5 P41594 3/20 0.40
GRM1 Q13255 2/20 0.40
MAPK1 P28482 1/20 0.40
DTYMK P23919 1/20 0.38
NAMPT P43490 1/20 0.37
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18181191 0.86 POLB (0.43) POLBGPR119GRM5GRM1MAPK1
SCHEMBL4598286 0.85 POLB (0.43) POLBGPR119GRM5GRM1MAPK1
SCHEMBL14097932 0.85 POLB (0.43) POLBGPR119GRM5GRM1MAPK1
SCHEMBL17094798 0.84 POLB (0.42) POLBGPR119GRM5GRM1MAPK1
SCHEMBL17094785 0.83 POLB (0.41) POLBGPR119GRM5GRM1MAPK1
SCHEMBL17094830 0.82 PTPN1 (0.42) POLBGPR119GRM5GRM1MAPK1
Lithium Ion SCHEMBL17094797 0.82 POLB (0.40) POLBGPR119GRM5GRM1MAPK1
SCHEMBL18181042 0.81 POLB (0.40) POLBGPR119GRM5GRM1MAPK1
SCHEMBL20024837 0.80 POLB (0.39) POLBGPR119GRM5GRM1MAPK1
SCHEMBL4597401 0.79 NR1D1 (0.40) POLBGPR119GRM5GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5681959-A DEPROTONATION OF A 2-AMINO-3-ALKYLPYRIDINE WITH AN ALKYLLITHIUM COMPOUND, THEN REACTION WITH AN AMIDE OR ESTER AND TREATMENT WITH A CONCENTRATED ACID FOR CYCLIZATION MERCK, SHARP & DOHME LTD. (GB) 1997-10-28 US disclosed