SCHEMBL8877698

SCHEMBL8877698

CCC(C(=O)Oc1c(-c2ccc(F)cc2)cc(-c2ccccc2)nc1C(C)C)(C(C)O)[PH](=O)OC

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 2/20 0.39
SQOR Q9Y6N5 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8879132 0.92 HMGCR (0.41) HMGCRSQORKDM4EALDH1A1LMNA
SCHEMBL8902033 0.90 HMGCR (0.34) HMGCRHPGD
SCHEMBL8877411 0.87 HMGCR (0.40) HMGCRSQOR
SCHEMBL8900012 0.84 DHODH (0.36)
SCHEMBL8877078 0.84 HMGCR (0.39) HMGCRSQORKDM4EALDH1A1LMNA
SCHEMBL8902222 0.83 GCGR (0.38)
SCHEMBL8877642 0.82 HMGCR (0.35) HMGCRHPGD
SCHEMBL8877739 0.79 HMGCR (0.41) HMGCRSQOR
SCHEMBL8878790 0.78 HMGCR (0.38) HMGCRSQORKDM4EALDH1A1LMNA
SCHEMBL8877505 0.78 HMGCR (0.40) HMGCRSQORKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed