SCHEMBL8877703

SCHEMBL8877703

CC(C)c1nc(C2CC2)cc(-c2ccc(F)cc2)c1C#COC(=O)CC(O)C[PH](=O)O

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
HMGCR P04035 1/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8877364 0.96 HMGCR (0.43) KDM4ENPSR1HTTL3MBTL1ADORA2A
SCHEMBL8877205 0.93 KDM4E (0.44) KDM4ENPSR1HTTL3MBTL1ADORA2A
SCHEMBL8878668 0.89 HMGCR (0.42) KDM4ENPSR1HTTL3MBTL1ADORA2A
SCHEMBL8877344 0.88 KDM4E (0.42) KDM4ENPSR1LMNAHPGD
SCHEMBL8876404 0.85
SCHEMBL8877297 0.84
SCHEMBL8876791 0.83
SCHEMBL8879853 0.83 ADORA3 (0.35) KDM4EL3MBTL1ADORA1MAPTHPGD
SCHEMBL8877068 0.81 KDM4E (0.41) KDM4ENPSR1LMNAHPGD
SCHEMBL8952905 0.80 NPSR1 (0.40) KDM4ENPSR1HTTL3MBTL1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed