SCHEMBL8877997

SCHEMBL8877997

COC(=O)CC(=O)c1ccc([N+](=O)[O-])cc1Cl

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.57
TDP1 Q9NUW8 2/20 0.57
MAPK1 P28482 2/20 0.56
GAA P10253 2/20 0.56
HTT P42858 2/20 0.56
NPSR1 Q6W5P4 1/20 0.56
MAPT P10636 6/20 0.53
POLB P06746 2/20 0.53
PKM P14618 1/20 0.52
NPC1 O15118 4/20 0.50
RAB9A P51151 4/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
MCL1 Q07820 1/20 0.50
ADRB2 P07550 1/20 0.50
ADRB1 P08588 1/20 0.50
ADRB3 P13945 1/20 0.50
FLT1 P17948 1/20 0.49
FLT4 P35916 1/20 0.49
KDR P35968 1/20 0.49
ALDH1A1 P00352 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11278115 0.88 TDP1 (0.57) KMT2ATDP1MAPK1GAAHTT
SCHEMBL28092969 0.82 KMT2A (0.64) KMT2ATDP1MAPK1GAAHTT
SCHEMBL222270 0.82 TDP1 (0.67) KMT2ATDP1MAPK1GAAHTT
SCHEMBL2223541 0.79 KMT2A (0.64) KMT2ATDP1MAPK1GAAHTT
SCHEMBL26215126 0.79 KMT2A (0.56) KMT2ATDP1MAPK1GAAHTT
SCHEMBL4372575 0.79 ERCC5 (0.63) KMT2ATDP1MAPK1MAPTPOLB
SCHEMBL1625685 0.78 MAPT (0.49) KMT2ATDP1MAPK1GAAHTT
SCHEMBL17690536 0.77 KMT2A (0.57) KMT2ATDP1MAPK1GAAHTT
SCHEMBL480106 0.77 KMT2A (0.70) KMT2ATDP1MAPK1GAAHTT
SCHEMBL7778630 0.76 MAPT (0.66) KMT2ATDP1GAAHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5672708-A Process for the preparation of N-arylaminoacrylic acid derivatives and the use of N-arylaminoacrylic acid derivatives thus prepared for the preparation of 4-quinolone-3-carboxylic acid derivatives BAYER AKTIENGESELLSCHAFT (DE) 1997-09-30 US disclosed