SCHEMBL8878033

SCHEMBL8878033

CC(C)c1nc(-c2c(F)c(F)cc(F)c2F)cc(-c2ccc(F)cc2)c1CO

nearest known ligand 0.55

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GCGR P47871 19/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6963687 0.82 GCGR (0.62) GCGR
SCHEMBL8877568 0.82 HMGCR (0.58) GCGR
SCHEMBL2663566 0.80 GCGR (0.58) GCGR
SCHEMBL8879625 0.79 HMGCR (0.44) GCGR
SCHEMBL8877443 0.79 GCGR (0.54) GCGR
SCHEMBL8876732 0.78 GCGR (0.44) GCGR
SCHEMBL8877373 0.77 GCGR (0.49) GCGR
SCHEMBL8877852 0.77 GCGR (0.49) GCGR
SCHEMBL8879135 0.76 GCGR (0.54) GCGR
SCHEMBL8949822 0.76 GCGR (0.88) GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed
US-5506219-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-04-09 US disclosed