SCHEMBL8878484

SCHEMBL8878484

C=C(C=O)c1c(-c2ccc(F)cc2)cc(-c2ccccc2)nc1C

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 2/20 0.45
SQOR Q9Y6N5 3/20 0.43
TOP1 P11387 2/20 0.42
ALDH1A1 P00352 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
DHODH Q02127 2/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
MAPT P10636 5/20 0.41
KDM4E B2RXH2 2/20 0.41
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
PTK2B Q14289 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8878404 0.84 HMGCR (0.48) HMGCRSQORTOP1DHODHADORA2A
SCHEMBL8878224 0.83 MAPT (0.51) HMGCRSQORTOP1ALDH1A1L3MBTL1
SCHEMBL8879664 0.78 HMGCR (0.54) HMGCRSQORTOP1ALDH1A1L3MBTL1
Pyridine SCHEMBL8878037 0.78 MAPT (0.46) HMGCRSQORTOP1ALDH1A1L3MBTL1
SCHEMBL8876854 0.76 HMGCR (0.48) HMGCRALDH1A1L3MBTL1DHODHMAPT
SCHEMBL8952895 0.75 HMGCR (0.55) HMGCRSQORTOP1ADORA2AADORA1
SCHEMBL8952886 0.75 HMGCR (0.55) HMGCRSQORTOP1ADORA2AADORA1
Methane SCHEMBL10345704 0.74 TOP1 (0.49) HMGCRSQORTOP1ALDH1A1L3MBTL1
SCHEMBL8878362 0.73 SQOR (0.48) HMGCRSQORTOP1ALDH1A1L3MBTL1
SCHEMBL8877552 0.70 MAPT (0.49) SQORTOP1DHODHADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed