SCHEMBL8879008

SCHEMBL8879008

C#CC(C(=O)Oc1c(C(C)C)nc(-c2ccccc2)c(C(C)C)c1-c1ccc(F)cc1)(C(C)O)[PH](=O)O

nearest known ligand 0.45

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 3/20 0.36
FABP4 P15090 2/20 0.33
GCGR P47871 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8876731 0.93 HMGCR (0.34) HMGCRGCGR
SCHEMBL8876603 0.93 HMGCR (0.34) HMGCRGCGR
SCHEMBL8901358 0.92 HMGCR (0.37) HMGCRGCGR
SCHEMBL8877422 0.92
SCHEMBL8876900 0.90 GCGR (0.38) GCGR
SCHEMBL8877856 0.86 HMGCR (0.37) HMGCRGCGR
SCHEMBL8899623 0.85 HMGCR (0.34) HMGCRGCGR
SCHEMBL8899571 0.85 HMGCR (0.34) HMGCRGCGR
SCHEMBL8878790 0.83 HMGCR (0.38) HMGCR
SCHEMBL8877114 0.83 HMGCR (0.52) HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed