SCHEMBL8879601

SCHEMBL8879601

COC(=O)C(Br)c1ccc(OCc2ccc3ccccc3n2)cc1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.59
CYSLTR1 Q9Y271 7/20 0.56
CYSLTR2 Q9NS75 5/20 0.56
PDE10A Q9Y233 4/20 0.56
ALOX5 P09917 4/20 0.56
HDAC6 Q9UBN7 1/20 0.56
FFAR1 O14842 1/20 0.55
AKR1B1 P15121 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7611388 0.88 GPBAR1 (0.62) GPBAR1CYSLTR1CYSLTR2PDE10AALOX5
SCHEMBL8648447 0.87 GPBAR1 (0.60) GPBAR1CYSLTR1CYSLTR2PDE10AALOX5
SCHEMBL9431747 0.86 GPBAR1 (0.59) GPBAR1CYSLTR1CYSLTR2PDE10AALOX5
SCHEMBL10410134 0.85 CYSLTR1 (0.58) GPBAR1CYSLTR1CYSLTR2PDE10AALOX5
SCHEMBL10410628 0.85 GPBAR1 (0.58) GPBAR1CYSLTR1CYSLTR2PDE10AALOX5
SCHEMBL8880806 0.83 CYSLTR1 (0.58) GPBAR1CYSLTR1CYSLTR2PDE10AALOX5
SCHEMBL10410185 0.83 GPBAR1 (0.56) GPBAR1CYSLTR1CYSLTR2PDE10AALOX5
SCHEMBL9498311 0.83 ALOX5 (0.54) GPBAR1CYSLTR1CYSLTR2PDE10AALOX5
SCHEMBL9589932 0.82 ALOX5 (0.66) GPBAR1CYSLTR1ALOX5
SCHEMBL7801682 0.82 ALOX5 (0.66) GPBAR1CYSLTR1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5597833-A LEUKOTRIENE SYNTHESIS INHIBITORS FOR ANTIINFLAMMATORY AGENTS, RESPIRATORY SYSTEM DISORDERS, ANTIALLERGENS OR ANTIISCHEMIC AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1997-01-28 US disclosed
CN-1087337-A The quinolin-2-ylmethoxy phenylacetic acid derivatives that replaces BAYER AG (DE) 1994-06-01 CN disclosed