SCHEMBL8879740

SCHEMBL8879740

O=C(CNCC(CCBr)c1ccc(Cl)cc1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RHOC P08134 10/20 0.43
RHOA P61586 10/20 0.43
UTS2R Q9UKP6 3/20 0.40
TACR1 P25103 1/20 0.39
P2RX1 P51575 1/20 0.38
CLPP Q16740 1/20 0.38
CNR2 P34972 1/20 0.37
PPARG P37231 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8069509 1.00 RHOC (0.43) RHOCRHOAUTS2RTACR1P2RX1
SCHEMBL8062563 0.90 TACR1 (0.39) TACR1
SCHEMBL8565826 0.89 MCHR1 (0.42) RHOCRHOAUTS2RTACR1
SCHEMBL8882416 0.89 MCHR1 (0.42) RHOCRHOAUTS2RTACR1
SCHEMBL8878961 0.83 UTS2R (0.37) UTS2R
SCHEMBL8559422 0.83 UTS2R (0.37) UTS2R
SCHEMBL8063644 0.80 TACR1 (0.43) TACR1
SCHEMBL8332703 0.76 TACR1 (0.56) RHOCRHOAUTS2RTACR1P2RX1
SCHEMBL8560072 0.75 MCHR1 (0.39) RHOCRHOATACR1P2RX1
SCHEMBL8560068 0.75 MCHR1 (0.39) RHOCRHOATACR1P2RX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607936-A USEFUL IN TREATMENT OF RESPIRATORY DISEASES MERCK & CO., INC. (US) 1997-03-04 US disclosed
WO-1996010568-A1 SUBSTITUTED ARYL PIPERAZINES AS NEUROKININ ANTAGONISTS MERCK & CO., INC. (US) 1996-04-11 WO disclosed