SCHEMBL8879744

SCHEMBL8879744

O=C(O)c1cn(C2CC2)c2c(OC(F)F)c(N3CCN(c4ccccc4)CC3)c(F)cc2c1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.56
KDM4E B2RXH2 8/20 0.56
ALDH1A1 P00352 5/20 0.56
HPGD P15428 4/20 0.56
POLB P06746 3/20 0.56
TDP1 Q9NUW8 2/20 0.56
OPRM1 P35372 2/20 0.56
HSD17B10 Q99714 2/20 0.56
PRKD3 O94806 1/20 0.56
ALOX15 P16050 1/20 0.56
CLK2 P49760 1/20 0.56
CLK4 Q9HAZ1 1/20 0.56
LMNA P02545 2/20 0.53
NPSR1 Q6W5P4 1/20 0.53
CHRM2 P08172 1/20 0.51
CHRM1 P11229 1/20 0.51
OPRD1 P41143 1/20 0.51
CYP2C19 P33261 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
MEN1 O00255 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27525623 0.91 KCNH2 (0.57) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL8879184 0.91 KCNH2 (0.59) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL8878712 0.89 KCNH2 (0.55) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL8880183 0.88 KCNH2 (0.57) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL7810777 0.87 KDM4E (0.64) KCNH2KDM4EALDH1A1HPGDPOLB
Hydrochloric Acid SCHEMBL8732413 0.87 KCNH2 (0.56) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL7813566 0.84 ALDH1A1 (0.73) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL6372074 0.83 KCNH2 (0.60) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL6372068 0.83 KCNH2 (0.60) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL8061803 0.83 ALDH1A1 (0.53) KCNH2KDM4EALDH1A1HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5519016-A Aryl group- or aromatic heterocyclic group-substituted aminoquinolone derivatives and anti-HIV agent UBE INDUSTRIES, LTD. (JP) 1996-05-21 US claimed
EP-0572259-A1 Aminoquinolone derivatives as anti-HIV agents UBE INDUSTRIES, LTD. (JP) 1993-12-01 EP claimed
US-5688791-A COMPOUNDS FOR TREATMENNT OF VIRAL DISEASES SUCH AS AIDS UBE INDUSTRIES, LTD. (JP) 1997-11-18 US disclosed
US-5519016-A Aryl group- or aromatic heterocyclic group-substituted aminoquinolone derivatives and anti-HIV agent UBE INDUSTRIES, LTD. (JP) 1996-05-21 US disclosed
EP-0572259-A1 Aminoquinolone derivatives as anti-HIV agents UBE INDUSTRIES, LTD. (JP) 1993-12-01 EP disclosed