SCHEMBL8880604

SCHEMBL8880604

Cc1cc(-c2nc3ccccc3c(C(C)C)c2C#CC(C(=O)O)(C(C)O)[PH](=O)O)ccc1F

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 2/20 0.36
DHODH Q02127 5/20 0.33
PDE10A Q9Y233 3/20 0.33
PRNP P04156 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
CTSA P10619 1/20 0.31
MAPK13 O15264 1/20 0.30
MAPK12 P53778 1/20 0.30
MAPK11 Q15759 1/20 0.30
MAPK14 Q16539 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8877820 0.79 HMGCR (0.41) HMGCRDHODHPDE10ACTSA
SCHEMBL8878936 0.79
SCHEMBL10345295 0.77 HMGCR (0.40) HMGCRCTSA
SCHEMBL8880612 0.77 HMGCR (0.39) HMGCRDHODHPDE10APRNPRXFP1
SCHEMBL8877812 0.74 PDE10A (0.33) HMGCRDHODHPDE10APRNPRXFP1
SCHEMBL8953516 0.73
SCHEMBL8953497 0.73
SCHEMBL8879913 0.71 HMGCR (0.34) HMGCR
SCHEMBL8877481 0.70
SCHEMBL8877788 0.69 PRNP (0.32) HMGCRPRNPRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed