SCHEMBL8880729

SCHEMBL8880729

NC(=O)C(CCC1CCCCN1)(c1ccccc1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.47
POLB P06746 1/20 0.46
CHRM3 P20309 8/20 0.43
CHRM2 P08172 6/20 0.43
CACNA2D1 P54289 1/20 0.42
CACNA1B Q00975 1/20 0.42
CACNB1 Q02641 1/20 0.42
CYP2D6 P10635 2/20 0.42
KCNH2 Q12809 2/20 0.42
LMNA P02545 1/20 0.42
CHRM1 P11229 1/20 0.42
KDM4E B2RXH2 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
HTR1A P08908 1/20 0.40
HTR1D P28221 1/20 0.40
HTR2A P28223 1/20 0.40
HRH1 P35367 1/20 0.40
ADRA1B P35368 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8879883 0.99 KMT2A (0.49) KMT2APOLBCHRM3CHRM2CACNA2D1
SCHEMBL1641984 0.79 POLB (0.51) KMT2APOLBCHRM3CHRM2CYP2D6
SCHEMBL8879197 0.73 KCNA3 (0.49) KMT2APOLBCHRM3CYP2D6KCNH2
SCHEMBL465843 0.73 POLB (0.48) KMT2APOLBCACNA2D1CACNA1BCACNB1
SCHEMBL22260272 0.72 CYP2D6 (0.48) KMT2APOLBCYP2D6LMNAKDM4E
SCHEMBL20833005 0.72 CYP2D6 (0.48) KMT2APOLBCYP2D6LMNAKDM4E
SCHEMBL6053465 0.72 POLB (0.47) KMT2APOLBCACNA2D1CACNA1BCACNB1
SCHEMBL678496 0.72 KDM4E (0.41) KMT2APOLBCHRM3CHRM2CYP2D6
SCHEMBL27886943 0.72 GHSR (0.42) KMT2APOLBCHRM3CYP2D6KDM4E
SCHEMBL27886944 0.72 GHSR (0.42) KMT2APOLBCHRM3CYP2D6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607950-A IRRITABLE BOWEL SYNDROME PFIZER INC. (US) 1997-03-04 US disclosed
EP-0508988-B1 MUSCARINIC RECEPTOR ANTAGONISTS PFIZER LTD (GB) 1994-03-02 EP disclosed
EP-0508988-A1 MUSCARINIC RECEPTOR ANTAGONISTS. PFIZER LTD (GB) 1992-10-21 EP disclosed
WO-1991010647-A1 MUSCARINIC RECEPTOR ANTAGONISTS PFIZER LIMITED (GB) 1991-07-25 WO disclosed