SCHEMBL8882

SCHEMBL8882

[c]1cnc2ccccc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
EGFR P00533 1/20 0.41
MAPT P10636 4/20 0.39
CYP1A2 P05177 2/20 0.39
HPGD P15428 3/20 0.39
GLA P06280 2/20 0.39
ACHE P22303 1/20 0.39
NQO2 P16083 2/20 0.37
KDM4E B2RXH2 3/20 0.37
GPR3 P46089 1/20 0.37
PDGFRB P09619 2/20 0.34
PDGFRA P16234 2/20 0.34
MGAM O43451 1/20 0.34
GAA P10253 2/20 0.33
HSD17B10 Q99714 2/20 0.33
NCF1 P14598 1/20 0.33
NOS2 P35228 1/20 0.33
BACE1 P56817 1/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6411133 0.98 ALDH1A1 (0.44) ALDH1A1EGFRMAPTCYP1A2HPGD
SCHEMBL27857176 0.98 ALDH1A1 (0.44) ALDH1A1EGFRMAPTCYP1A2HPGD
SCHEMBL27765897 0.96 ALDH1A1 (0.43) ALDH1A1EGFRMAPTCYP1A2HPGD
SCHEMBL17511856 0.80 NQO2 (0.43) ALDH1A1MAPTCYP1A2HPGDGLA
SCHEMBL452574 0.76
SCHEMBL21858493 0.76 ALDH1A1 (0.50) ALDH1A1MAPTCYP1A2HPGDGLA
SCHEMBL451496 0.74
SCHEMBL695179 0.74 BACE1 (0.42) PDGFRBPDGFRAGAABACE1TDP1
SCHEMBL4657766 0.74 ALDH1A1 (0.50) ALDH1A1MAPTCYP1A2NQO2KDM4E
SCHEMBL9481501 0.73 CYP3A4 (0.55) ALDH1A1MAPTKDM4EGPR3HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 27372 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4392032-A1 MODULATORS OF THE BETA-3 ADRENERGIC RECEPTOR FOR THE TREATMENT OR PREVENTION OF RENAL CYSTIC DISEASE AND CARDIORENAL SYNDROME Arena Pharmaceuticals, Inc. (US) 2024-07-03 EP claimed
CN-118267472-A Naphthopin cation derivative and application thereof in biological medicine and material field 上海先辉医药科技有限公司 2024-07-02 CN claimed
US-20240208927-A1 WNT SIGNALING PATHWAY INHIBITORS FOR TREATMENTS OF DISEASE UNIVERSITY OF MARYLAND, BALTIMORE 2024-06-27 US claimed
CN-118221579-A PRMT5 inhibitors 北京望实智慧科技有限公司 2024-06-21 CN claimed
US-20240199604-A1 SUPRAMOLECULAR POLYMER THERAPEUTICS AND DIAGNOSTICS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-06-20 US claimed
US-20240197682-A1 METHOD FOR TREATING NEUROLOGICAL DISEASES USING SUPRAMOLECULE POLYMER THERAPEUTICS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-06-20 US claimed
US-20240201205-A1 METHOD FOR DETECTING NEUROLOGICAL DISEASES USING SUPRAMOLECULE POLYMER THERAPEUTICS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-06-20 US claimed
WO-2024108147-A1 COMPOUNDS, COMPOSITIONS, AND METHODS DENALI THERAPEUTICS INC. (US) 2024-05-23 WO claimed
US-11987588-B2 Modulators of the beta-3 adrenergic receptor useful for the treatment or prevention of heart failure and disorders related thereto ARENA PHARMACEUTICALS, INC. (US) 2024-05-21 US claimed
US-20240156792-A1 COMBINATION THERAPY USING AZABICYCLO COMPOUND FOR CANCER TAIHO PHARMACEUTICAL CO., LTD. (JP) 2024-05-16 US claimed
US-4385058-A HISTAMINE H2-ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1983-05-24 US claimed
US-4379154-A Thiocarboxamide derivatives and their use as pharmaceuticals RHONE-POULENC SANTE (FR) 1983-04-05 US claimed
EP-0049173-A2 Pyrimidone derivatives, processes for their preparation and pharmaceutical derivatives containing them SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1982-04-07 EP claimed
EP-0047109-A1 Rhodanine derivatives, process for their preparation, and aldose reductase inhibitor containing the rhodanine derivatives as active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 1982-03-10 EP claimed
EP-0003677-B1 PYRIMIDONES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1981-11-11 EP claimed
EP-0003677-A2 Pyrimidones, processes for their preparation and pharmaceutical compositions containing them SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-08-22 EP claimed
US-4163784-A ACYLUREA DERIVATIVES PFIZER INC. (US) 1979-08-07 US claimed
US-3993645-A Stilbene optical brighteners and compositions brightened therewith STERLING DRUG INC. (US) 1976-11-23 US claimed
US-3968102-A VASODILATOR, ANTICOAGULANT KOHJIN CO., LTD. (JA) 1976-07-06 US claimed
US-3932301-A NYLON, POLYESTERS STERLING DRUG INC. (US) 1976-01-13 US claimed