SCHEMBL8884091

SCHEMBL8884091

CC(C)Oc1cccc(C(=O)N2CC[C@](CCOS(C)(=O)=O)(c3cccc4ccccc34)C2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
HTT P42858 2/20 0.47
GAA P10253 1/20 0.47
TACR2 P21452 3/20 0.39
TACR1 P25103 3/20 0.39
KCNK3 O14649 1/20 0.38
KCNK9 Q9NPC2 1/20 0.38
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
LMNA P02545 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
USP2 O75604 1/20 0.38
TP53 P04637 1/20 0.38
PKM P14618 2/20 0.37
PKLR P30613 1/20 0.35
POLB P06746 2/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9028736 0.94 MEN1 (0.52) MEN1KMT2AHTTGAATACR2
SCHEMBL8884481 0.88 MEN1 (0.47) MEN1KMT2AHTTGAATACR2
SCHEMBL8883531 0.87 TACR2 (0.48) TACR2TACR1
SCHEMBL9027155 0.82 MEN1 (0.52) MEN1KMT2AHTTGAATACR2
SCHEMBL8883877 0.79 KMT2A (0.46) MEN1KMT2AHTTGAATACR2
SCHEMBL8883870 0.79 KMT2A (0.46) MEN1KMT2AHTTGAATACR2
SCHEMBL9028740 0.77 KDM4E (0.39) MEN1KMT2AHTTGAAALDH1A1
SCHEMBL8884449 0.76 TACR2 (0.55) MEN1KMT2ATACR2TACR1
SCHEMBL9027244 0.75 KMT2A (0.47) MEN1KMT2AHTTGAATACR2
SCHEMBL6990563 0.74 TACR2 (0.47) GAATACR2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607947-A Pyrrolidinyl tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1997-03-04 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed