SCHEMBL8884615

SCHEMBL8884615

CS(=O)(=O)OCC[C@]1(c2cccc(Cl)c2)CCN(C(=O)Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)C1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 13/20 0.45
OPRK1 P41145 2/20 0.43
OPRD1 P41143 1/20 0.43
CNR1 P21554 1/20 0.41
TACR2 P21452 2/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
EPHX2 P34913 1/20 0.39
SLC6A4 P31645 1/20 0.38
KCNH2 Q12809 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9028652 0.95 EPHX2 (0.44) TACR1OPRK1OPRD1CNR1MEN1
SCHEMBL9027567 0.94 MEN1 (0.43) TACR1OPRK1OPRD1CNR1MEN1
SCHEMBL8883694 0.90 TACR1 (0.46) TACR1OPRK1OPRD1CNR1TACR2
SCHEMBL8882055 0.90 TACR1 (0.46) TACR1OPRK1OPRD1CNR1TACR2
SCHEMBL8883348 0.89 TACR1 (0.42) TACR1OPRK1OPRD1CNR1TACR2
SCHEMBL8884286 0.87 TACR1 (0.42) TACR1OPRK1OPRD1CNR1TACR2
SCHEMBL8884315 0.87 TACR1 (0.42) TACR1OPRK1OPRD1CNR1TACR2
SCHEMBL8884136 0.87 TACR1 (0.45) TACR1OPRK1OPRD1CNR1TACR2
SCHEMBL8883296 0.86 TACR1 (0.41) TACR1OPRK1OPRD1CNR1TACR2
SCHEMBL8882764 0.86 TACR1 (0.41) TACR1OPRK1OPRD1CNR1TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607947-A Pyrrolidinyl tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1997-03-04 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed