SCHEMBL8889407

SCHEMBL8889407

COc1ccc(CCCc2cc(C(=O)Nc3c(Cl)cncc3Cl)ccc2OC)cc1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 12/20 0.62
PDE4B Q07343 12/20 0.61
PDE4A P27815 9/20 0.61
PDE4C Q08493 9/20 0.61
CYP2B6 P20813 1/20 0.55
P2RX7 Q99572 1/20 0.50
HTR1D P28221 1/20 0.46
HTR1B P28222 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890987 0.89 PDE4D (0.66) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8891532 0.85 PDE4D (0.66) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8891122 0.82 PDE4D (0.62) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8890532 0.79 PDE4D (0.70) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL30614148 0.79 PDE4D (0.68) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8892506 0.78 PDE4B (0.76) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL15270505 0.78 PDE4D (1.00) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8888978 0.78 PDE4D (0.65) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8890369 0.77 PDE4B (0.74) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8890145 0.77 PDE4D (0.61) PDE4DPDE4BPDE4APDE4CCYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO claimed
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO disclosed