SCHEMBL8891532

SCHEMBL8891532

COc1ccc(C(=O)Nc2c(Cl)cncc2Cl)cc1CCc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 17/20 0.66
PDE4A P27815 15/20 0.59
PDE4B Q07343 15/20 0.59
PDE4C Q08493 15/20 0.59
CYP2B6 P20813 1/20 0.58
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
GFER P55789 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8889907 0.88 PDE4D (0.64) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL8891152 0.87 PDE4D (0.62) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL8890145 0.86 PDE4D (0.61) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL8889648 0.85 PDE4B (0.74) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL8889407 0.85 PDE4D (0.62) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL8888978 0.84 PDE4D (0.65) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL8890369 0.84 PDE4B (0.74) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL8889614 0.83 PDE4D (0.73) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL6948901 0.83 PDE4B (0.73) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL8890987 0.81 PDE4D (0.66) PDE4DPDE4APDE4BPDE4CCYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO claimed
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO disclosed