SCHEMBL8889477

SCHEMBL8889477

Cc1cc(N2C(=O)CN(Cc3ccccc3)CC2=O)ccc1OCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.46
FFAR4 Q5NUL3 1/20 0.45
MAPK14 Q16539 2/20 0.43
MEN1 O00255 5/20 0.42
KMT2A Q03164 5/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MRGPRX4 Q96LA9 2/20 0.40
S1PR5 Q9H228 1/20 0.40
MCHR1 Q99705 1/20 0.40
PTGER1 P34995 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
REV1 Q9UBZ9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7358848 0.80 SNRNP200 (0.51) MAPK14MEN1KMT2ANPC1RAB9A
SCHEMBL9080839 0.79 DRD4 (0.55) MEN1KMT2ANPC1RAB9AMAPK1
SCHEMBL8915218 0.72 FFAR4 (0.46) FFAR4NPC1RAB9AMRGPRX4MCHR1
SCHEMBL3143366 0.71 FFAR4 (0.44) FFAR4MAPK14NPC1RAB9AMAPK1
SCHEMBL3135075 0.71 FFAR4 (0.44) FFAR4MEN1KMT2ANPC1RAB9A
SCHEMBL11527905 0.70 CYP3A4 (0.45) CYP3A4MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL1101974 0.70 MC4R (0.53) MEN1KMT2ANPC1RAB9AMAPK1
Hydrochloric Acid SCHEMBL8888785 0.69 HTR1A (0.61) FFAR4MRGPRX4
SCHEMBL13144443 0.69 MRGPRX4 (0.68) FFAR4MEN1KMT2ANPC1RAB9A
SCHEMBL4720449 0.68 MAPK14 (0.52) MAPK14MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652242-A 3-METHYL-4-(4-(4-(4-PYRIDYL)PIPERAZIN-1-YL)PHENOXY)BURYIC ACID, AMIDE OR ESTER; INHIBITORS OF BINDING OF FIBRINOGEN TO GLYCOPROTEIN ZENECA LIMITED (GB) 1997-07-29 US disclosed
US-5563141-A INHIBIT CELL ADHESION FOR EXAMPLE, PLATELET AGGRE GATION ZENECA LIMITED (GB) 1996-10-08 US disclosed