SCHEMBL8890705

SCHEMBL8890705

COc1cccc(Nc2nc(Nc3ccc(C#N)cc3)nc3ccccc23)c1

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 3/20 0.67
ABCG2 Q9UNQ0 12/20 0.64
KDM4E B2RXH2 1/20 0.60
HTT P42858 1/20 0.60
TAAR1 Q96RJ0 1/20 0.60
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
ABCB1 P08183 5/20 0.58
PDE5A O76074 1/20 0.58
MERTK Q12866 2/20 0.57
RXFP1 Q9HBX9 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8889951 0.99 NPY5R (0.66) NPY5RABCG2KDM4EHTTTAAR1
SCHEMBL8891851 0.90 NPY5R (0.78) NPY5RABCG2KDM4EHTTTAAR1
Hydrochloric Acid SCHEMBL8890746 0.89 NPY5R (0.77) NPY5RABCG2HTTTAAR1MEN1
Hydrochloric Acid SCHEMBL8899399 0.89 NPY5R (0.76) NPY5RABCG2KDM4EHTTTAAR1
SCHEMBL8889167 0.89 NPY5R (0.76) NPY5RABCG2KDM4EHTTTAAR1
Hydrochloric Acid SCHEMBL8907334 0.88 NPY5R (0.83) NPY5RABCG2KDM4EHTTTAAR1
Hydrochloric Acid SCHEMBL8907425 0.88 HTT (0.75) NPY5RABCG2KDM4EHTTTAAR1
SCHEMBL8898863 0.86 NPY5R (0.74) NPY5RABCG2KDM4EMEN1KMT2A
SCHEMBL8891079 0.86 NPY5R (0.72) NPY5RABCG2KDM4EHTTTAAR1
Hydrochloric Acid SCHEMBL8890523 0.85 NPY5R (0.72) NPY5RABCG2KDM4EHTTTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed