SCHEMBL8891017

SCHEMBL8891017

CCS(=O)(=O)Cc1ccc(Nc2nc(NC3CC3)c3cccc(OC)c3n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 2/20 0.53
MERTK Q12866 6/20 0.50
PDE5A O76074 3/20 0.44
HDAC1 Q13547 3/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC3 O15379 1/20 0.40
DNMT1 P26358 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
DNMT3A Q9Y6K1 1/20 0.40
USP2 O75604 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
DAPK3 O43293 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8890172 0.99 NPY5R (0.52) NPY5RMERTKPDE5AHDAC1HDAC6
SCHEMBL8891826 0.86 NPY5R (0.71) NPY5RMERTK
Hydrochloric Acid SCHEMBL8889262 0.85 NPY5R (0.70) NPY5RMERTK
SCHEMBL8890639 0.79 MERTK (0.63) NPY5RMERTKUSP2CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL8901180 0.78 MERTK (0.62) NPY5RMERTKUSP2CYP1A2CYP3A4
SCHEMBL8892661 0.76 MERTK (0.56) MERTK
SCHEMBL8899654 0.75 NPY5R (0.56) NPY5RMERTK
SCHEMBL8890967 0.75 NPY5R (0.74) NPY5R
Hydrochloric Acid SCHEMBL8890483 0.75 MERTK (0.56) MERTK
SCHEMBL8891020 0.75 PDE5A (0.40) MERTKPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed