SCHEMBL8891545

SCHEMBL8891545

COc1ccc(F)cc1[C@@]1(O)[C@H](O)CC(c2ccccc2)(c2ccccc2)[C@@H]2CN(C(=O)C(CCCc3ccccc3)N(C)C)C[C@@H]21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.44
LPAR1 Q92633 3/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
HPGD P15428 2/20 0.32
HTR2A P28223 3/20 0.32
HTR2C P28335 3/20 0.32
HTR2B P41595 2/20 0.32
NR3C1 P04150 1/20 0.32
MC4R P32245 1/20 0.32
MC5R P33032 1/20 0.32
MC1R Q01726 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
CACNA1F O60840 1/20 0.32
DRD1 P21728 1/20 0.32
DRD4 P21917 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8890811 0.99 TACR1 (0.44) TACR1LPAR1FNTAFNTBSIGMAR1
Bromide SCHEMBL8890169 0.91 TACR1 (0.41) TACR1LPAR1SIGMAR1HPGD
SCHEMBL8891566 0.82 TACR1 (0.41) TACR1FNTAFNTBHTR2AHTR2C
Bromide SCHEMBL8890843 0.81 TACR1 (0.41) TACR1FNTAFNTBHTR2AHTR2C
SCHEMBL8890274 0.81 TACR1 (0.42) TACR1FNTAFNTB
Bromide SCHEMBL8891352 0.79 TACR1 (0.41) TACR1FNTAFNTB
SCHEMBL8891554 0.78 TACR1 (0.39) TACR1FNTAFNTBHTR2AHTR2C
Bromide SCHEMBL8890819 0.77 TACR1 (0.39) TACR1FNTAFNTBHTR2AHTR2C
Bromide SCHEMBL8890180 0.73 TACR1 (0.38) TACR1FNTAFNTBOPRD1OPRK1
SCHEMBL8548123 0.73 TACR1 (0.73) TACR1FNTAFNTBHPGDADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997005110-A1 PERHYDROISOINDOLE DERIVATIVES AS SUBSTANCE P AND NEUROKININE A ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1997-02-13 WO claimed
WO-1997005110-A1 PERHYDROISOINDOLE DERIVATIVES AS SUBSTANCE P AND NEUROKININE A ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1997-02-13 WO disclosed