SCHEMBL8891554

SCHEMBL8891554

COc1ccc(F)cc1[C@@]1(O)[C@H](O)CC(c2ccccc2)(c2ccccc2)[C@@H]2CN(C(=O)CCC[N+](C)(C)Cc3ccccc3)C[C@@H]21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.39
FNTA P49354 2/20 0.37
FNTB P49356 2/20 0.37
BCHE P06276 2/20 0.35
ACHE P22303 2/20 0.35
MC4R P32245 2/20 0.33
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
MC5R P33032 1/20 0.33
MC1R Q01726 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CACNA1F O60840 1/20 0.33
DRD1 P21728 1/20 0.33
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33
HRH2 P25021 1/20 0.33
ADRA1D P25100 1/20 0.33
HTR7 P34969 1/20 0.33
ADRA1A P35348 1/20 0.33
HRH1 P35367 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8890819 0.99 TACR1 (0.39) TACR1FNTAFNTBBCHEACHE
Bromide SCHEMBL8890170 0.91 ALDH1A1 (0.37) TACR1FNTAFNTBBCHEACHE
SCHEMBL8890828 0.87 TACR1 (0.33) TACR1FNTAFNTBBCHEACHE
SCHEMBL8890274 0.85 TACR1 (0.42) TACR1FNTAFNTBBCHEACHE
SCHEMBL8891566 0.82 TACR1 (0.41) TACR1FNTAFNTBMC4RHTR2A
Bromide SCHEMBL8890843 0.81 TACR1 (0.41) TACR1FNTAFNTBMC4RHTR2A
Bromide SCHEMBL8891355 0.80 ALDH1A1 (0.38) TACR1FNTAFNTBBCHEACHE
SCHEMBL8890176 0.79 KDM4E (0.34) TACR1FNTAFNTBACHE
SCHEMBL8891545 0.78 TACR1 (0.44) TACR1FNTAFNTBMC4RHTR2A
Bromide SCHEMBL8890811 0.77 TACR1 (0.44) TACR1FNTAFNTBMC4RHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997005110-A1 PERHYDROISOINDOLE DERIVATIVES AS SUBSTANCE P AND NEUROKININE A ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1997-02-13 WO claimed
WO-1997005110-A1 PERHYDROISOINDOLE DERIVATIVES AS SUBSTANCE P AND NEUROKININE A ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1997-02-13 WO disclosed