SCHEMBL8892003

SCHEMBL8892003

Cc1ccc(C(=O)Nc2c(Cl)cncc2Cl)cc1OC(C)c1ccccn1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 13/20 0.53
PDE4B Q07343 13/20 0.48
PDE4A P27815 7/20 0.48
PDE4C Q08493 7/20 0.48
NOX1 Q9Y5S8 3/20 0.48
CYP2B6 P20813 1/20 0.47
ABCB11 O95342 1/20 0.46
BRD4 O60885 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890302 0.79 BRD4 (0.47) NOX1BRD4
SCHEMBL8891475 0.79 BRD4 (0.47) NOX1BRD4
SCHEMBL8892009 0.78 PDE4D (0.55) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL15920428 0.72 PDE4D (0.71) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8888975 0.72 PDE4D (0.70) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL7353637 0.71 PDE4D (0.81) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL7361933 0.71 PDE4D (0.76) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL7421279 0.71 PDE4D (0.78) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL6874729 0.70 PDE4D (0.81) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL15270505 0.70 PDE4D (1.00) PDE4DPDE4BPDE4APDE4CCYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO claimed
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO disclosed