SCHEMBL8893337

SCHEMBL8893337

CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)[C@@H]1C[C@@H](Cc2ccc(C(F)(F)F)cc2)C(=O)O1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
ATM Q13315 1/20 0.40
CTSS P25774 3/20 0.39
CTSK P43235 2/20 0.39
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
ACE P12821 1/20 0.38
SCN9A Q15858 2/20 0.38
KMT2A Q03164 1/20 0.38
AKT1 P31749 1/20 0.37
REN P00797 1/20 0.37
MAPK1 P28482 1/20 0.37
ALDH1A1 P00352 1/20 0.37
APP P05067 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8892992 0.96 PPARG (0.41) PPARGPPARAATMCTSSCTSK
SCHEMBL8892378 0.96 PPARG (0.41) PPARGPPARAATMCTSSCTSK
SCHEMBL8893594 0.93 CTSS (0.41) PPARGPPARAATMCTSSCTSK
SCHEMBL7426423 0.93 CTSS (0.41) PPARGPPARAATMCTSSCTSK
SCHEMBL8893975 0.93 CTSS (0.41) PPARGPPARAATMCTSSCTSK
SCHEMBL7443701 0.93 ATM (0.46) ATMCTSSCTSKCTSLCTSB
SCHEMBL6312228 0.93 ATM (0.46) ATMCTSSCTSKCTSLCTSB
SCHEMBL7432732 0.93 ATM (0.46) ATMCTSSCTSKCTSLCTSB
SCHEMBL9005035 0.93 ATM (0.46) ATMCTSSCTSKCTSLCTSB
SCHEMBL6786029 0.91 CTSS (0.45) ATMCTSSCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643878-A TREATMENT OF RETROVIRAL DISEASES LIKE AIDS CIBA-GEIGY CORPORATION (US) 1997-07-01 US disclosed
WO-1996016980-A1 MORPHOLINOETHYLAMIDE DERIVATIVES NOVARTIS AG (CH) 1996-06-06 WO disclosed
EP-0618222-A2 Dipeptid derivatives of 5-amino-4-hydroxy-hexanoic acid CIBA-GEIGY AG (CH) 1994-10-05 EP disclosed