SCHEMBL8895878

SCHEMBL8895878

CN1CCN(c2ncc(-c3cc(F)c(Cl)c(Cl)c3Cl)c(N)n2)CC1

nearest known ligand 0.69

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNK2 O95069 1/20 0.69
SCN2A Q99250 1/20 0.69
PTPN11 Q06124 8/20 0.47
HTR3A P46098 2/20 0.44
HRH4 Q9H3N8 3/20 0.43
KMT2A Q03164 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
BCL6 P41182 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8902764 0.85 KCNK2 (0.56) KCNK2SCN2APTPN11HTR3AHRH4
Sipatrigine SCHEMBL29421474 0.81 SCN2A (1.00) KCNK2SCN2APTPN11HTR3AHRH4
Sipatrigine SCHEMBL135888 0.81 SCN2A (1.00) KCNK2SCN2APTPN11HTR3AHRH4
SCHEMBL7282208 0.80 KCNK2 (0.71) KCNK2SCN2APTPN11HTR3AHRH4
SCHEMBL7272345 0.77 KCNK2 (0.71) KCNK2SCN2APTPN11HTR3AHRH4
SCHEMBL8895638 0.77 KCNK2 (0.60) KCNK2SCN2APTPN11HTR3AHRH4
SCHEMBL5070764 0.77 KCNK2 (0.74) KCNK2SCN2APTPN11HTR3AHRH4
Sipatrigine SCHEMBL5069235 0.75 SCN2A (0.85) KCNK2SCN2APTPN11HTR3AHRH4
SCHEMBL8894121 0.74 DHFR (0.47) KCNK2SCN2A
SCHEMBL12922468 0.74 KCNK2 (0.60) KCNK2SCN2APTPN11HTR3AHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020827-A1 FLUOROPHENYL-TRIAZINE AND PYRIMIDINE DERIVATIVES AS COMPOUNDS ACTING ON THE CENTRAL NERVOUS SYSTEM LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 1997-06-12 WO claimed