SCHEMBL8895977

SCHEMBL8895977

Cc1nc(N)c(C#N)nc1-c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.42
CTSK P43235 3/20 0.42
IKBKB O14920 2/20 0.41
XDH P47989 3/20 0.40
SLC9A5 Q14940 1/20 0.35
USP8 P40818 1/20 0.35
MBOAT4 Q96T53 1/20 0.34
ADORA2A P29274 3/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
BRD4 O60885 1/20 0.33
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
ADORA1 P30542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8898393 0.75 ATR (0.44) CTSSCTSKIKBKBXDHALDH1A1
SCHEMBL11370778 0.74 CHEK1 (0.53) USP8ADORA2AALDH1A1MEN1KMT2A
SCHEMBL11368597 0.72 ERBB2 (0.47) IKBKBUSP8ADORA2AALDH1A1MEN1
SCHEMBL8896372 0.72 CTSS (0.46) CTSSCTSKIKBKBXDHADORA2A
SCHEMBL8898622 0.70 PIK3CG (0.43) IKBKBALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL28823040 0.69 DPP4 (0.51) USP8ADORA2AALDH1A1MEN1KMT2A
SCHEMBL10087551 0.68 HSD17B10 (0.38) USP8ADORA2AALDH1A1
SCHEMBL11809427 0.68 CHEK1 (0.53) USP8ADORA2AALDH1A1MEN1KMT2A
SCHEMBL21722354 0.65 ADORA2A (0.58) ADORA2AALDH1A1MEN1KMT2AADORA1
SCHEMBL8649829 0.65 IKBKB (0.40) CTSSCTSKIKBKBXDHADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639753-A CONTROLLING INSECTS IN AGRICULTURE CROPS FMC CORPORATION (US) 1997-06-17 US disclosed
US-5532367-A LARVICIDES FMC CORPORATION (US) 1996-07-02 US disclosed
US-5521190-A USEFUL AGAINST TOBACCO BUDWORM FMC CORPORATION (US) 1996-05-28 US disclosed
WO-1994027439-A1 INSECTICIDAL PTERIDINES AND 8-DEAZAPTERIDINES FMC CORPORATION (US) 1994-12-08 WO disclosed